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PAPERS PUBLISHED

  1. Makarov, M.; Sanchez Rocha, A.C.; Krystufek, R.; Cherepashuk, I.; Dzmitruk, V.; Charnavets, T.; Faustino, A.M; Lebl, M.; Fujishima, K.; Fried, S.D.; Hlouchova, K. Early selection of the amino acid alphabet was adaptively shaped by biophysical constraints of foldability . J.Am.Chem.Soc. 2023, 145, 5320–5329. 2023JACS_5320.pdf

  2. Lebl, M. How to make sure that you will get the Nobel Prize . Chem. Listy 2023, 117 , 485–486. 2023ChemListy.pdf

  3. Pazderkova, M.; Bednarova, L.; Dlouha, H.; Lebl, M.; Hlavacek, J.; Setnicka, V.; Urbanova, M.; Hynie, S.; Klenerova, V.; Baumruk, V.; Malon, P.. Electronic and vibrational optical activity of several peptides related to neurohypophyseal hormones: Disulfide group conformation. Biopolymers 2012, 97 , 923–932. 2012Biopolymers.pdf

  4. Lebl-Rinnova, M.; Tran, H. N.; Lebl, M. Modified synthesis of safety catch acid-labile (SCAL) linker. In: Peptides, Building Bridges: The Proceedings of The Twenty-Second American Peptide Symposium, Lebl, M., Ed.; Prompt Scientific Publishing: San Diego, 2011; pp 40-41. 2011Proc22APS_40.pdf

  5. Lebl, M.; Heiner, D.; Jones, A. C.; Fambro, S. P.; Nibbe, M. J.; Burgett, S. R.; Ellman, B. M. Automatic oligonucleotide synthesizer utilizing the concept of parallel processing. Collection Symposium Series 2011, 12, 264-267. 2011CCCC.pdf

  6. Lebl, M.; Slaninova, J. Ala-Walk analogs of oxytocin - HPLC-based conformational studies. In: Peptides, Building Bridges: The Proceedings of The Twenty-Second American Peptide Symposium, Lebl, M., Ed.; Prompt Scientific Publishing: San Diego, 2011; pp 316-317. 2011Proc22APS_316.pdf

  7. Lebl, M. Combinatorial/Library Peptide Synthesis. In: Amino Acids, Peptides and Proteins in Organic Chemistry, Hughes, A. B., Ed.; Wiley: Weinheim, 2011; pp 395-449. 2011AAPeptProt.pdf

  8. Schroeder, M. A.; Salloum, K. S.; Perbost, M.; Lebl, M.; Posner, J. D. Radial flow electroosmotic pump. Sensor. Actuator. A-Phys. 2011, 169 (1), 250-255. 2011SensorsActuators.pdf

  9. Kozlov, I. A.; Melnyk, P. C.; Hachmann, J. P.; Srinivasan, A.; Shults, M. D.; Zhao, C.; Musmacker, J.; Nelson, N.; Barker, D. L.; Lebl, M. A high-complexity, multiplexed solution-phase assay for profiling protease activity on microarrays. Comb. Chem. High Throughput Screening 2008, 11, 24-35. 2008CombChemHighThrScr.pdf

  10. Remacle, A. G.; Shiryaev, S. A.; Oh, E. S.; Cieplak, P.; Srinivasan, A.; Wei, G.; Liddington, R. C.; Ratnikov, B. I.; Parent, A.; Desjardins, R.; Day, R.; Smith, J. W.; Lebl, M.; Strongin, A. Y. Substrate cleavage analysis of furin and related proprotein convertases. Journal of Biological Chemistry 2008, 283 (30), 20897-20906. 2008JBiolChem.pdf

  11. Kermani, B. G.; Kozlov, I. A.; Melnyk, P. C.; Zhao, C.; Hachmann, J. P.; Lebl, M. Using support vector machine regression to model the retention of peptides in immobilized metal-affinity chromatography. Sensors. and Actuators B: Chemical 2007, 125, 149-157. 2007SensActBChem.pdf

  12. Kozlov, I. A.; Kermani, B. G.; Melnyk, P. C.; Barker, D. L.; Zhao, C.; Hachmann, J. P.; Lebl, M. Study of the retention of histidine containing peptides on nickel column. J. Chromatogr. Sci. 2007, 45, 207-211. span style="text-decoration: underline;">2007JChromSci.pdf

  13. Kozlov, I. A.; Melnyk, P. C.; Hachmann, J. P.; Barker, D. L.; Lebl, M.; Zhao, C. Evaluation of different chemical strategies for conjugation of oligonucleotides to peptides. Nucleosides, Nucleotides & Nucleic Acids 2007, 26 (10), 1353-1357. 2007NuclNuclNuclAcids.pdf

  14. Lebl, M.; Kozlov, I. A.; Melnyk, P. C.; Hachmann, J. P.; Srinivasan, A.; Shults, M. D.; Musmacker, J.; Nelson, N.; Kermani, B. G.; Zhao, C.; Barker, D. L. High complexity protease and kinase profiling solution assays with readout on randomly assembled microarrays. In: Proc.29th Eur. Pept. Symp., Gdansk, 2006, 2007; p in press. 2007Proc29EPS.pdf

  15. Lebl, M.; Pistek, C.; Hachmann, J. P.; Mudra, P.; Pesek, V.; Pokorny, V.; Poncar, P.; Zenisek, K. Economical parallel oligonucleotide and peptide synthesizer - Pet Oligator. International Journal of Peptide Research and Therapeutics 2007, 13 (1-2), 367-375. 2007IntJPeptResTherap.pdf

  16. Raman, B.; Kotseroglou, T.; Clark, L.; Lebl, M.; Gutierrez-Osuna, R. Neuromorphic processing for optical microbead arrays: dimensionality reduction and contrast enhancement. IEEE Sensors Journal 2007, 7 (4), 506-514. 2007IEEESensorsJournal.pdf

  17. Shiryaev, S. A.; Kozlov, I. A.; Ratnikov, B. I.; Smith, J. W.; Lebl, M.; Strongin, A. Y. Cleavage preference distinguishes the two-component NS2B-NS3 serine proteinases of Dengue and West Nile viruses. Biochem. J. 2007, 401, 743-752. 2007BiochemJ.pdf

  18. Shiryaev, S. A.; Ratnikov, B. I.; Aleshin, A. E.; Kozlov, I. A.; Nelson, N. A.; Lebl, M.; Smith, J. W.; Liddington, R. C.; Strongin, A. Y. Switching the substrate specificity of the two-component NS2B-NS3 flaviviral proteinase by structure-based mutagenesis. J. Virol. 2007, 81 (9), 4501-4509. 2007JVirology.pdf

  19. Shiryaev, S. A.; Remacle, A. G.; Ratnikov, B. I.; Nelson, N. A.; Savinov, A. Y.; Wei, G.; Bottini, M.; Rega, M. F.; Parent, A.; Desjardins, R.; Fugere, M.; Day, R.; Sabet, M.; Pellecchia, M.; Liddington, R. C.; Smith, J. W.; Mustelin, T.; Guiney, D. G.; Lebl, M.; Strongin, A. Y. Targeting host cell furin proprotein convertases as a therapeutic strategy against bacterial toxins and viral pathogens. Journal of Biological Chemistry 2007, 282 (29), 20847-20853. 2007JBiolChem.pdf

  20. Shults, M. D.; Kozlov, I. A.; Nelson, N.; Kermani, B. G.; Melnyk, P. C.; Shevchenko, V.; Srinivasan, A.; Musmacker, J.; Hachmann, J. P.; Barker, D. L.; Lebl, M.; Zhao, C. A multiplexed protein kinase assay. Chembiochem 2007, 8, 933-942. 2007ChemBiochem.pdf

  21. Hachmann, J. P.; Lebl, M. Alternative to piperidine in Fmoc solid phase synthesis. J. Comb. Chem. 2006, 8, 149. 2006JCombChem.pdf

  22. Hachmann, J. P.; Lebl, M. Search for optimal coupling reagent in multiple peptide synthesizer. Biopolymers (Pept. Sci. ) 2006, 84, 340-347. 2006Biopolymers.pdf

  23. Hachmann, J. P.; Lebl, M. Synthesis of poly d(G-C) oligonucleotides. Nucleosides, Nucleotides and Nucleic Acids 2006, 25 (7), 705-717. 2006NuclNuclNuclAcids.pdf

  24. Kermani, B. G.; Fomenko, I.; Kotseroglou, T.; Forood, B.; Clark, L.; Barker, D.; Lebl, M. Decoding beads in a randomly assembled optical nose. Sensors and Actuators B 2006, 117, 282-285. 2006SensorsActuatorsB.pdf

  25. Kozlov, I. A.; Melnyk, P. C.; Zhao, C.; Hachmann, J. P.; Shevchenko, V.; Srinivasan, A.; Barker, D. L.; Lebl, M. A method for rapid protease substrate evaluation and optimization. Comb. Chem. High Throughput Screening 2006, 9, 481-487. 2006CombChemHighThrScr.pdf

  26. Lebl, M.; Barker, D. L.; Kozlov, I. A.; Melnyk, P. C.; Hachmann, J. P.; Srinivasan, A.; Shults, M.; Nelson, N.; Zhao, C. Multiplexed profiling of protease and kinase substrate with readout on oligonucleotide microarrays. J. Peptide Sci. 2006, 12, 95. WOS:000239905600053

  27. Lebl, M.; Hachmann, J. P. High-throughput peptide synthesis. Howl, J., Ed.; Humana Press, Inc.: Totowa, NJ, 2005; pp 167-194. 2005MethMolBiol.pdf

  28. Lebl, M. Combinatorial chemistry. In: Encyclopedia of 20th-Century Technology, Hempstead, C. A., Worthington, W. E., Eds.; Routledge: New York, 2005; pp 171-174. 2005Encyclopedia20thCentTechnol.pdf

  29. Lebl, M.; Pokorny, V.; Krchnak, V. Simple tools for resin distribution. J. Comb. Chem. 2005, 7, 42-45. 2005JCombChem.pdf

  30. Kermani, B.; Fomenko, I.; Kotseroglou, T.; Forood, B.; Clark, L.; Barker, D.; Lebl, M. Supervised learning for decoding beads in a randomly-assembled optical nose. In: Computational Biology Workshop, Neural Information Processing System (NIPS), 11th Annual Conference, Whistler, BC, Canada, 2004. 2002ONosePosters.pdf

  31. Kermani, B.; Kotseroglou, T.; Forood, B.; Barker, D.; Lebl, M. Optical nose signal denoising and detrending using wavelets. In: Proceedings of 8th World Multiconference on Systems, Cybernetics, and Informatics, Orlando, FL, 2004; pp 148-149. 2002ONosePosters.pdf

  32. Lebl, M. Centrifugation based automated synthesis technologies. J. Assoc. Lab. Autom. 2003, 8 (3), 30-36. 2003JALA.pdf

  33. Forood, B.; Kotseroglou, T.; Clark, L.; Lebl, M.; Lieu, M.-H.; Kermani, B.; Barker, D.; Dickinson, T. Chemical detection using Illumina's BeadArray technology. In: Proc. 9th International Symposium on Olfaction and Electronic Nose, ISOEN'02, Rome, 2002. 2002ONosePosters.pdf

  34. Lam, K. S.; Lebl, M. Synthesis of one-bead-one-compound combinatorial peptide library. In: Protein Protocols on CD-ROM Version 2.0, John M.Walker, Ed.; Humana Press: Totowa, NJ, 2002; pp 20-24. 2002ProtProtocolsCD.pdf

  35. Lebl, M. Combinatorial chemistry: The history and the basics. In: Integrated Drug Discovery Technologies; 2002. 2002IntegrDrugDiscTechnol.pdf

  36. Lebl, M.; Pires, J.; Burger, C.; Ni, Y.; Chen, Y. Solid-phase parallel synthesis of large tetrahydroisoquinolinone library. In: High-Throughput Synthesis, Sucholeiki, I., Ed.; Marcel Dekker, Inc.: New York, 2001; pp 187-195. 2001HighThrSynt_187.pdf

  37. Lebl, M.; Burger, C.; Ellman, B.; Heiner, D.; Ibrahim, G.; Jones, A.; Nibbe, M.; Thompson, J.; Mudra, P.; Pokorny, V.; Poncar, P.; Zenisek, K. Fully automated parallel oligonucleotide synthesizer. Collect. Czech. Chem. Commun. 2001, 66, 1299-1314. 2001CCCC.pdf

  38. Lebl, M.; Pires, J. Solid-phase parallel synthesis of a large array of tetrahydroisoquinolinones. In: High-Throughput Synthesis, Sucholeiki, I., Ed.; Marcel Dekker, Inc.: New York, 2001; pp 197-205. 2001HighThrSynt_197.pdf

  39. Lebl, M.; Houghten, R. A. Preface. In: Peptides; The Wave of the Future. Proc. 2nd Int. 17th Amer. Pept. Symp.; Lebl, M., Houghten, R. A., Eds.; American Peptide Society: San Diego, 2001; p ix-xi. 2001Proc17APS.pdf

  40. Lebl, M.; Burger, C.; Ellman, B.; Heiner, D.; Ibrahim, G.; Jones, A.; Nibbe, M.; Pires, J.; Mudra, P.; Pokorny, V.; Poncar, P.; Zenisek, K. Fully automated parallel oligonucleotide synthesizer. In: Peptides; The Wave of the Future. Proc. 2nd Int. 17th Amer. Pept. Symp.; Lebl, M., Houghten, R. A., Eds.; American Peptide Society: San Diego, 2001; pp 277-278. 2001Proc17APS_277.pdf

  41. Eichler, J.; Lebl, M. Combinatorial chemistry: A powerful tool for basic research and drug discovery. Journal of Clinical Ligand Assay 2000, 23 (4), 262-272. 2000JClinLigAssay.pdf

  42. Eichler, J.; Lebl, M. La chimica combinatoria: un potente strumento per la ricerca di base e la ricerca farmacologica. Journal of Clinical Ligand Assay 2000, 23, 262-272. 2000JCLA_Italian.pdf

  43. Lebl, M.; Ma, J.; Pires, J.; Dooley, C.; Houghten, R. A. Rapid parallel synthesis of 584 betides, peptides composed largely of beta-amino acids with side-chains not found in natural peptides. In: Peptides for the New Millennium, Fields, G. B., Tam, J. P., Barany, G., Eds.; Kluwer Academic Publisher: Dordrecht, 2000; pp 174-175. 1999Proc16APS_174.pdf

  44. Lebl, M. New technique for high-throughput synthesis of peptides, peptidomimetics and nonpeptide small organic molecule arrrays. In: Peptides for the New Millennium, Fields, G. B., Tam, J. P., Barany, G., Eds.; Kluwer Academic Publisher: Dordrecht, 2000; pp 164-166. 1999Proc16APS_164.pdf

  45. Ni, Y.; Krchnak, V.; Lebl, M. New approach for preparation of 2,3,7-trisubstituted 3,4-dihydroisoquinolinone libraries on solid phase. Mol. Diversity 2000, 5 (3), 153-161. 2000MolDiv.pdf

  46. Lebl, M. New approaches to automatic synthesis of large arrays of small organic molecules. In: Proceedings of combinatorial chemistry conference; Osaka, Japan, 1999; pp 6-14. 1999ProcOsaka.pdf

  47. Lebl, M.; Pires, J.; Poncar, P.; Pokorny, V. Evaluation of gaseous hydrogen fluoride as a convenient reagent for parallel cleavage from the solid support. J. Comb. Chem. 1999, 1 (6), 474-479. 1999JCombChem_474.pdf

  48. Lebl, M. Sooner or later someone else will cotton on to this idea (in " Matrix Assisted Synthetic Transformations: A Mosaic of Diverse Contributions. II. The Pattern Is Completed" by D. Hudson). J. Comb. Chem. 1999, 1 (6), 438-442. 1999JCombChem_403.pdf

  49. Lebl, M. New technique for high-throughput synthesis. Bioorg. Med. Chem. Lett. 1999, 9 (9), 1305-1310. 1999BioorgMedChemLett.pdf

  50. Lebl, M. Parallel personal comments on "classical" papers in combinatorial chemistry. J. Comb. Chem. 1999, 1 (1), 3-24. 1999JCombChem_003.pdf

  51. Lebl, M.; Krchnak, V.; Ibrahim, G.; Pires, J.; Burger, C.; Ni, Y.; Chen, Y.; Podue, D.; Mudra, P.; Pokorny, V.; Poncar, P.; Zenisek, K. Solid-phase synthesis of large tetrahydroisoquinolinone arrays by two different approaches. Synthesis-Stuttgart 1999, (11), 1971-1978. 1999Synthesis.pdf

  52. Lebl, M.; Krchnak, V. Techniques for massively parallel synthesis of small organic molecules. In: Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries, Epton, R., Ed.; Mayflower Scientific Limited: Birmingham, 1999; pp 43-46. 1998InnovPerspSPS_043.pdf

  53. Lebl, M. Solid-phase synthesis of combinatorial libraries. Curr. Opin. Drug. Disc. Develop. 1999, 2 (4), 385-395. 1999CurrOpinDrugDiscDev.pdf

  54. Rinnova, M.; Lebl, M.; Soucek, M. Solid-phase peptide synthesis by fragment condensation: Coupling in swelling volume. Lett. Peptide Sci. 1999, 6, 15-22. 1999LettPeptSci.pdf

  55. Rinnova, M.; Soucek, M.; Voburka, Z.; Lebl, M.; Fusek, M. Sanger's reagent: An excellent end-capping and/or labeling agent for SPPS. In: Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries, Epton, R., Ed.; Mayflower Scientific Limited: Birmingham, 1999; pp 385-386. 1998InnovPerspSPS_385.pdf

  56. Thorpe, D. S.; Yeoman, H.; Chan, A. W. E.; Krchnak, V.; Lebl, M.; Felder, S. Combinatorial chemistry reveals a new motif that binds the platelet fibrinogen receptor, gpIIbIIIa. Biochem. Biophys. Res. Commun. 1999, 256 (3), 537-541. 1999BiochemBiophyResComm.pdf

  57. Lam, K. S.; Lebl, M. Synthesis of a one-bead one-compound combinatorial peptide library. Methods in Molecular Biology (Totowa, New Jersey) 1998, 87 (Combinatorial Peptide Library Protocols), 1-6. 1998CombPeptLibProt.pdf

  58. Lebl, M. Solid-phase synthesis on planar supports. Biopolymers (Pept. Sci. ) 1998, 47 (5), 397-404. 1998PeptSci_397.pdf

  59. Lebl, M. A new approach to automated solid phase synthesis based on centrifugation of tilted plates. J. Assoc. Lab. Autom. 1998, 3 (3), 59-61. 1998JALA.pdf

  60. Ostrem, J. A.; Al-Obeidi, F.; Safar, P.; Safarova, A.; Stringer, S. K.; Patek, M.; Cross, M. T.; Spoonamore, J.; LoCascio, J. C.; Kasireddy, P.; Thorpe, D. S.; Sepetov, N.; Lebl, M.; Wildgoose, P.; Strop, P. Discovery of a novel, potent, and specific family of factor Xa inhibitors via combinatorial chemistry. Biochemistry 1998, 37 (4), 1053-1059. 1998Biochemistry.pdf

  61. Patek, M.; Lebl, M. Safety-catch and multiply cleavable linkers in solid-phase synthesis. Biopolymers (Pept. Sci. ) 1998, 47 (5), 353-363. 1998PeptSci_353.pdf

  62. Seligmann, B.; Lebl, M.; Lam, K. S. Solid-phase peptide synthesis, lead generation, and optimization. In: Combinatorial Chemistry and Molecular Diversity in Drug Discovery, Gordon, E. M., Kerwin, J. F. J., Eds.; John Wiley & Sons: New York, 1998; pp 39-109. 1998CombChemMolDivDrugDisc.pdf

  63. Cargill, J. F.; Lebl, M. New methods in combinatorial chemistry: Robotics and parallel synthesis. Curr. Opin. Chem. Biol. 1997, 1 (1), 67-71. 1997CurrOpinChemBiol.pdf

  64. Krchnak, V.; Weichsel, A. S.; Lebl, M.; Felder, S. Automated solid-phase organic synthesis in micro-plate wells. Synthesis of N-(alkoxy-acyl)amino alcohols. Bioorg. Med. Chem. Lett. 1997, 7 (8), 1013-1016. 1997BioorgMedChemLett.pdf

  65. Lam, K. S.; Lebl, M.; Krchnak, V. The "one-bead-one-compound" combinatorial library method. Chem. Rev. 1997, 97 (2), 411-448. 1997ChemRev.pdf

  66. Lebl, M.; Krchnak, V. Synthetic peptide libraries. Methods Enzymol. 1997, 289, 336-392. 1997MethEnzymol.pdf

  67. Chen, C. L.; Strop, P.; Lebl, M.; Lam, K. S. One bead-one compound combinatorial peptide library: Different types of screening. Methods Enzymol. 1996, 267, 211-219. 1996MethEnzymol.pdf

  68. Eichler, J.; Houghten, R. A.; Lebl, M. Inclusion volume solid-phase peptide synthesis. J. Peptide Sci. 1996, 2 (4), 240-244. 1996JPeptSci.pdf

  69. Hruby, V. J.; Shenderovich, M.; Lam, K. S.; Lebl, M. Design considerations and computer modeling related to the development of molecular scaffolds and peptide mimetics for combinatorial chemistry. Mol. Diversity 1996, 2 (1-2), 46-56. 1996MolDiv_46.pdf

  70. Krchnak, V.; Weichsel, A. S.; Cabel, D.; Lebl, M. Structurally homogenous and heterogenous libraries: Scaffold- based libraries and libraries built using bifunctional building blocks. In: Molecular Diversity and Combinatorial Chemistry. Libraries and Drug Discovery, Chaiken, I. M., Janda, K. D., Eds.; American Chemical Society: Washington,DC, 1996; pp 99-117. 1996MolDivCombChem.pdf

  71. Krchnak, V.; Vagner, J.; Flegelova, Z.; Weichsel, A. S.; Barany, G.; Lebl, M. Use of solid-phase Mitsunobu and Wittig reactions for contruction of peptide and non-peptide libraries. In: Peptides:Chemistry,Structure and Biology,Proc.14.APS, Kaumaya, P. T. P., Hodges, R. S., Eds.; Mayflower Scientific Ltd.: Kingswinford, 1996; pp 307-308. 1996Proc14APS_307.pdf

  72. Krchnak, V.; Lebl, M. MARS: Multiple automatic robot synthesizer featuring a novel timing procedure and random access to reagents and reaction vessels. In: Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries, Epton, R., Ed.; Mayflower Scientific Limited: Birmingham, 1996; pp 93-96. 1996InnovPerspSPS_093.pdf

  73. Krchnak, V.; Sepetov, N. F.; Kocis, P.; Patek, M.; Lam, K. S.; Lebl, M. Combinatorial libraries of synthetic structures: Synthesis, screening, and structure determination. In: Combinatorial Libraries: Synthesis, Screening and Application Potential, Cortese, R., Ed.; Walter de Gruyter: Berlin, 1996; pp 27-52. 1996CombLib_Cortese.pdf

  74. Krchnak, V.; Weichsel, A. S.; Cabel, D.; Flegelova, Z.; Lebl, M. Structurally homogenous and heterogenous synthetic combinatorial libraries. Mol. Diversity 1996, 1 (3), 149-164. 1995MolDiv_149.pdf

  75. Krchnak, V.; Lebl, M. Synthetic library techniques: Subjective (biased and generic) thoughts and views. Mol. Diversity 1996, 1 (3), 193-216. 1995MolDiv_193.pdf

  76. Krchnak, V.; Cabel, D.; Lebl, M. MARS: Multiple automated robotic synthesizer for continuous flow of peptides. Peptide Res. 1996, 9 (1), 45-49. 1996PeptRes_45.pdf

  77. Lam, K. S.; Lou, Q.; Zhao, Z. G.; Chen, M. L.; Salmon, S. E.; Wade, S.; Lebl, M. Identification and applications of idiotype-specific peptides for two murine B-cell lymphoma cell lines. In: Peptides:Chemistry,Structure and Biology,Proc.14.APS, Kaumaya, P. T. P., Hodges, R. S., Eds.; Mayflower Scientific Ltd.: Kingswinford, 1996; pp 806-807. 1996Proc14APS_806.pdf

  78. Lam, K. S.; Lebl, M. Combinatorial library based on the one-bead-one-compound concept. In: Combinatorial Peptide and Nonpeptide Libraries: A Handbook, Jung, G., Ed.; VCH: Weinheim, 1996; pp 173-201. 1996CombPeptNonpeptLibraries.pdf

  79. Lam, K. S.; Lake, D.; Salmon, S. E.; Smith, J.; Chen, M. L.; Wade, S.; Abdul-Latif, F.; Leblova, Z.; Ferguson, R. D.; Krchnak, V.; Sepetov, N. F.; Lebl, M. A one-bead one-peptide combinatorial library method for B-cell epitope mapping. Methods: A Companion to Methods in Enzymology 1996, 9, 482-493. 1996Methods_482.pdf

  80. Lebl, M.; Krchnak, V.; Strop, P.; Lam, K. S. Construction and screening of peptide and nonpeptide libraries based on one-bead-one-compound principle. In: Peptides:Chemistry,Structure and Biology,Proc.14.APS, Kaumaya, P. T. P., Hodges, R. S., Eds.; Mayflower Scientific Ltd.: Kingswinford, 1996; pp 890-892. 1996Proc14APS_890.pdf

  81. Lebl, M.; Krchnak, V.; Patek, M.; Lam, K. S. Synthetic combinatorial libraries of scaffolded and unordered structures. Methods Mol. Cell. Biol. 1996, 6 (1), 41-55. 1995MethMolCellBiol_41.pdf

  82. Rinnova, M.; Fusek, M.; Lebl, M. Use of methyl red in solid phase synthesis. In: Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries, Epton, R., Ed.; Mayflower Scientific Limited: Birmingham, 1996; pp 509-510. 1996InnovPerspSPS_509.pdf

  83. Rinnova, M.; Lebl, M. Molecular diversity and libraries of structures: Synthesis and screening. Collect. Czech. Chem. Commun. 1996, 61, 171-231. 1996CCCC_0171.pdf

  84. Salmon, S. E.; Liu-Stevens, R. H.; Zhao, Y.; Lebl, M.; Krchnak, V.; Wertman, K.; Sepetov, N.; Lam, K. S. High-volume cellular screening for anticancer agents with combinatorial chemical libraries: A new methodology. Mol. Diversity 1996, 2 (1-2), 57-63. 1996MolDiv_57.pdf

  85. Stankova, M.; Lebl, M. Library generation through successive substitution of trichlorotriazine. Mol. Diversity 1996, 2 (1-2), 75-80. 1996MolDiv_75.pdf

  86. Stankova, M.; Strop, P.; Chen, C.; Lebl, M. Mixtures of molecules versus mixtures of pure compounds on polymeric beads. In: Molecular Diversity and Combinatorial Chemistry. Libraries and Drug Discovery, Chaiken, I. M., Janda, K. D., Eds.; American Chemical Society: Washington,DC, 1996; pp 137-143. 1996MolDivCombChem.pdf

  87. Vagner, J.; Krchnak, V.; Lebl, M.; Barany, G. Solid-phase organic synthesis: Creation of carbon-carbon double bond under mild conditions by Wittig-type reactions. Collect. Czech. Chem. Commun. 1996, 61, 1697-1702. 1996CCCC_1697.pdf

  88. Vagner, J.; Barany, G.; Lam, K. S.; Krchnak, V.; Sepetov, N. F.; Ostrem, J. A.; Strop, P.; Lebl, M. Enzyme-mediated spatial segregation on individual polymeric support beads: Application to generation and screening of encoded combinatorial libraries. Proc. Natl. Acad. Sci. USA 1996, 93 (16), 8194-8199. 1996PNAS_Vagner.pdf

  89. Flegelova, Z.; Krchnak, V.; Sepetov, N. F.; Stankova, M.; Issakova, O.; Cabel, D.; Lam, K. S.; Lebl, M. Libraries of small compact structures based on N-acyl-N-alkylamino acids. In: Peptides 94, Proc.23.EPS, Maia, H. L. S., Ed.; ESCOM: Leiden, 1995; pp 469-470. 1995Proc23EPS_469.pdf

  90. Geysen, H. M.; Houghten, R. A.; Kauffman, S.; Lebl, M.; Moos, W. H.; Pavia, M. R.; Szostak, J. W. Molecular diversity comes of age. Mol. Diversity 1995, 1 (1), 1-3. 1995MolDiv_001.pdf

  91. Kasal, A.; Kohout, L.; Lebl, M. Synthesis of a scaffold for the creation of non-peptide libraries. Collect. Czech. Chem. Commun. 1995, 60, 2147-2155. 1995CCCC_2147.pdf

  92. Kocis, P.; Issakova, O.; Sepetov, N. F.; Lebl, M. Kemp's triacid scaffolding for synthesis of combinatorial nonpeptide uncoded libraries. Tetrahedron Lett. 1995, 36, 6623-6626. 1995TetLett_6623.pdf

  93. Krchnak, V.; Weichsel, A. S.; Cabel, D.; Lebl, M. Linear presentation of variable side-chain spacing in a highly diverse combinatorial library. Peptide Res. 1995, 8 (4), 198-205. 1995PeptRes_198.pdf

  94. Krchnak, V.; Weichsel, A. S.; Issakova, O.; Lam, K. S.; Lebl, M. Bifunctional scaffolds as templates for synthetic combinatorial libraries. Mol. Diversity 1995, 1 (3), 177-182. 1995MolDiv_177.pdf

  95. Krchnak, V.; Flegelova, Z.; Weichsel, A. S.; Lebl, M. Polymer-supported Mitsunobu ether formation and its use in combinatorial chemistry. Tetrahedron Lett. 1995, 36, 6193-6196. 1995TetLett_6193.pdf

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  112. Lam, K. S.; Lebl, M. Selectide technology: Bead-binding screening. Methods: A Companion to Methods in Enzymology 1994, 6, 372-380. 1994Methods_372.pdf

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  120. Madden, D.; Krchnak, V.; Lebl, M. Synthetic combinatorial libraries: Views on techniques and their application. Perspect. Drug Disc. Design 1994, 2, 269-286. 1994PerspDrugDiscDes.pdf

  121. Majer, P.; Slaninova, J.; Lebl, M. Synthesis of methylated phenylalanines via hydrogenolysis of corresponding 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acids. Int. J. Peptide Prot. Res. 1994, 43 (1), 62-68. 1994IntJPeptProtRes_62.pdf

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  123. Patek, M.; Drake, B.; Lebl, M. All-cis cyclopentane scaffolding for combinatorial solid phase synthesis of small non-peptide compounds. Tetrahedron Lett. 1994, 35 (49), 9169-9172. 1994TetLett.pdf

  124. Pokorny, V.; Mudra, P.; Jehnicka, J.; Zenisek, K.; Pavlik, M.; Voburka, Z.; Rinnova, M.; Stierandova, A.; Lucka, A. W.; Eichler, J.; Houghten, R. A.; Lebl, M. Compas 242. New type of multiple peptide synthesizer utilizing cotton and tea bag technology. In: Innovation and Perspectives in Solid Phase Synthesis, Epton, R., Ed.; Mayflower Worldwide Limited: Birmingham, 1994; pp 643-648. 1994InnovPerspSPS_643.pdf

  125. Prochazka, Z.; Slaninova, J.; Melin, P.; Aurell, C. J.; Lebl, M. The deamino-carba analogs of vasotocin. Synthesis and some biological properties. Collect. Czech. Chem. Commun. 1994, 59, 421-428. 1994CCCC_0421.pdf

  126. Safar, P.; Slaninova, J.; Lebl, M. The carba-modification of cystine-containing peptides: Synthesis of selectively protected cystathionines and their incorporation into the oxytocin molecule. In: Peptides: Chemistry, Structure and Biology,Proc.13.APS, Hodges, R. S., Smith, J. A., Eds.; ESCOM: Leiden, 1994; pp 119-120. 1994Proc13APS_119.pdf

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  129. Sepetov, N. F.; Issakova, O. L.; Lebl, M.; Swiderek, K.; Stahl, D. C.; Lee, T. D. Hydrogen-deuterium exchange as a method facilitating unambiguous assignment of fragment ions in CID spectra of peptides. In: Peptides: Chemistry, Structure and Biology,Proc.13.APS, Hodges, R. S., Smith, J. A., Eds.; ESCOM: Leiden, 1994; pp 259-261. 1994Proc13APS_259.pdf

  130. Smith, M. H.; Lam, K. S.; Hersh, E. M.; Lebl, M.; Grimes, W. J. Peptide sequences binding to MHC class I proteins. Mol. Immunol. 1994, 31 (18), 1431-1437. 1994MolImmunol.pdf

  131. Stankova, M.; Wade, S.; Lam, K. S.; Lebl, M. Synthesis of combinatorial libraries with only one representation of each structure. Peptide Res. 1994, 7 (6), 292-298. 1994PeptRes_292.pdf

  132. Stankova, M.; Issakova, O.; Sepetov, N. F.; Krchnak, V.; Lam, K. S.; Lebl, M. Application of one-bead one-structure approach to identification of nonpeptidic ligands. Drug Develop. Res. 1994, 33, 146-156. 1994DrugDevRes_146.pdf

  133. Stierandova, A.; Sepetov, N. F.; Nikiforovich, G. V.; Lebl, M. Sequence-dependent modification of Trp by the Pmc protecting group of Arg during TFA deprotection. Int. J. Peptide Prot. Res. 1994, 43 (1), 31-38. 1994IntJPeptProtRes_31.pdf

  134. Vagner, J.; Krchnak, V.; Sepetov, N. F.; Strop, P.; Lam, K. S.; Barany, G.; Lebl, M. Novel methodology for differentiation of "surface" and "interior" areas of poly(oxyethylene)-polystyrene (POE-PS) supports: Application to library screening procedures. In: Innovation and Perspectives in Solid Phase Synthesis, Epton, R., Ed.; Mayflower Worldwide Limited: Birmingham, 1994; pp 347-352. 1994InnovPerspSPS_347.pdf

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  144. Munson, M. C.; Lebl, M.; Slaninova, J.; Barany, M. Solid-phase synthesis and biological activity of the parallel dimer of deamino-oxytocin. Peptide Res. 1993, 6 (3), 155-160. 1993PeptRes_155.pdf

  145. Nikolaiev, V.; Stierandova, A.; Krchnak, V.; Seligmann, B.; Lam, K. S.; Salmon, S. E.; Lebl, M. Peptide-encoding for structure determination of nonsequenceable polymers within libraries synthesized and tested on solid-phase supports. Peptide Res. 1993, 6 (3), 161-170. 1993PeptRes_161.pdf

  146. Prochazka, Z.; Zertova, M.; Slaninova, J.; Barth, T.; Majer, P.; Lebl, M. The new 8-D-homoarginine-vasopressin analogs with strong in vitro and in vivo uterus inhibiting activity. In: Peptides 1992, Proc.22.EPS, Schneider, C. H., Eberle, A. N., Eds.; ESCOM: Leiden, 1993; pp 717-718. 1993Proc22EPS_717.pdf

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  148. Rinnova, M.; Jezek, J.; Malon, P.; Lebl, M. Comparative multiple synthesis of fifty linear peptides: Evaluation of cotton carrier vs T bag-benzhydrylamine resin. Peptide Res. 1993, 6 (2), 88-94. 1993PeptRes_088.pdf

  149. Salmon, S. E.; Lam, K. S.; Lebl, M.; Kandola, A.; Khattri, P. S.; Wade, S.; Patek, M.; Kocis, P.; Krchnak, V.; Thorpe, D.; Felder, S. Discovery of biologically active peptides in random libraries: Solution-phase testing after staged orthogonal release from resin beads. Proc. Natl. Acad. Sci. USA 1993, 90 (24), 11708-11712. 1993PNAS_Salmon.pdf

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  151. Stahl, D. C.; Lee, T. D.; Sepetov, N. F.; Issakova, O. L.; Lebl, M. Computer program for interpreting peptide mass spectra utilizing hydrogen-deuterium exchange information. <None Specified> . 1993. Proceedings of 41.ASMS Conference on Mass Spectroscopy and Allied Topics, May 31-Lune 4, San Francisco, 1993. 1654 1993ProcASMS.pdf

  152. Zertova, M.; Prochazka, Z.; Slaninova, J.; Barth, T.; Majer, P.; Lebl, M. The analogs of [D-Har(8)]vasopressin with di- and trisubstituted phenylalanine in position 2; synthesis and some biological properties. Collect. Czech. Chem. Commun. 1993, 58, 2751-2760. 1993CCCC_2751.pdf

  153. Fric, I.; Lebl, M.; Hruby, V. J. Melanin concentrating hormone analogs : Contraction of the cyclic structure. III. CD spectroscopic study. Collect. Czech. Chem. Commun. 1992, 57, 614-620. 1992CCCC_0614.pdf

  154. Jezek, R.; Franc, J.; Slaninova, J.; Lebl, M. Sequence modification in neurohypophyseal hormones. Collect. Czech. Chem. Commun. 1992, 57, 621-624. 1992CCCC_0621.pdf

  155. Lam, K. S.; Lebl, M. Streptavidin and avidin recognize peptide ligands with different motifs. Immunomethods 1992, 1, 11-15. 1992Immunomethods.pdf

  156. Lebl, M.; Stierandova, A.; Eichler, J.; Patek, M.; Pokorny, V.; Jehnicka, J.; Mudra, P.; Zenisek, K.; Kalousek, J. An automated multiple solid phase peptide synthesizer utilizing cotton as a carrier. In: Innovation and Perspectives in Solid Phase Peptide Synthesis, Epton, R., Ed.; Intercept Limited: Andover, 1992; pp 251-257. 1992InnovPerspSPS_251.pdf

  157. Lebl, M.; Toth, G.; Slaninova, J.; Hruby, V. J. Conformationally biased analogs of oxytocin. Int. J. Peptide Prot. Res. 1992, 40 (2), 148-151. 1992IntJPeptProtRes_148.pdf

  158. Matsunaga, T. O.; Hruby, V. J.; Lebl, M.; Castrucci, A. M. L.; Hadley, M. E. Synthesis and bioactivity studies of two isosteric acyclic analogues of melanin concentrating hormone. Life Sci. 1992, 51 (9), 679-685. 1992LifeSci.pdf

  159. Pal, B. C.; Slaninova, J.; Barth, T.; Trojnar, J.; Lebl, M. Synthesis and properties of "hormonogene" and "inhibitorogene" type oxytocin analogs. Collect. Czech. Chem. Commun. 1992, 57, 1345-1351. 1992CCCC_1345.pdf

  160. Patek, M.; Lebl, M. Safety-catch protecting groups in peptide synthesis. Collect. Czech. Chem. Commun. 1992, 57, 508-524. 1992CCCC_0508.pdf

  161. Patek, M.; Lebl, M.; Budesinsky, M. Unusual KF/Al2O3 promoted tandem electrophilic-nucleophilic aromatic substitution leading to the xanthone formation. Tetrahedron Lett. 1992, 33, 4507-4508. 1992TetLett.pdf

  162. Prochazka, Z.; Slaninova, J.; Barth, T.; Stierandova, A.; Trojnar, J.; Melin, P.; Lebl, M. Analogs of deamino carba oxytocin with inhibitory properties; synthesis and some biological properties. Collect. Czech. Chem. Commun. 1992, 57, 1335-1344. 1992CCCC_1335.pdf

  163. Tourwe, D.; Toth, G.; Lebl, M.; Verschueren, K.; Knapp, R. J.; Davis, P.; Van Binst, G.; Yamamura, H. I.; Burks, T. K.; Kramer, T.; Hruby, V. J. A simple synthesis of 1,2,3,4-tetrahydro-7-hydroxyisoquinoline-3-carboxylic acid (HO-Tic) a conformationally constrained tyrosine analog and its incorporation into opioid peptides. In: Peptides: Chemistry and Biology, Proc.12.APS, Smith, J. A., Rivier, J. E., Eds.; ESCOM: Leiden, 1992; pp 307-308. 1992Proc12APS_307.pdf

  164. Verschueren, K.; Toth, G.; Tourwe, D.; Lebl, M.; Van Binst, G.; Hruby, V. J. Facile synthesis of 1,2,3,4-tetrahydro-7-hydroxyisoquinoline-3-carboxylic acid, a conformationally constrained tyrosine analogue. Synthesis-Stuttgart 1992, 458-460. 1992Synthesis.pdf

  165. Zertova, M.; Prochazka, Z.; Slaninova, J.; Barth, T.; Lebl, M. Amino and deamino analogs of 8-D-homoarginin-vasopressin with modified tyrosine in position 2: Synthesis and some biological properties. Collect. Czech. Chem. Commun. 1992, 57, 604-613. 1992CCCC_0604.pdf

  166. Zertova, M.; Prochazka, Z.; Slaninova, J.; Barth, T.; Majer, P.; Lebl, M. The analogs of 8-D-homoarginin-vasopressin with o-substituted phenylalanine in position 2: Synthesis and some biological properties. Collect. Czech. Chem. Commun. 1992, 57, 1103-1110. 1992CCCC_1103.pdf

  167. Cerovsky, V.; Safar, P.; Prochazka, Z.; Lebl, M. Papain-catalyzed selective incorporation of cystathionine derivatives into model peptides. In: Peptides 90, Proc.21.EPS, Giralt, E., Andreu, D., Eds.; ESCOM: Leiden, 1991; pp 305-306. 1991Proc21EPS_305.pdf

  168. Eichler, J.; Furkert, J.; Bienert, M.; Rohde, W.; Lebl, M. Multiple peptide synthesis on cotton carriers: Elucidation and characterization of an antibody binding site of CRF. In: Peptides 90, Proc.21.EPS, Giralt, E., Andreu, D., Eds.; ESCOM: Leiden, 1991; pp 156-157. 1991Proc21EPS_156.pdf

  169. Eichler, J.; Bienert, M.; Stierandova, A.; Lebl, M. Evaluation of cotton as a carrier for solid phase peptide synthesis. Peptide Res. 1991, 4 (5), 296-307. 1991PeptRes_296.pdf

  170. Hilgert, I.; Stolba, P.; Kristofova, H.; Stefanova, I.; Bendlova, B.; Lebl, M.; Horejsi, V. A monoclonal antibody applicable for determination of C-peptide of human proinsulin by RIA. Hybridoma 1991, 10 (3), 379-386. 1991Hybridoma.pdf

  171. Lebl, M.; Fang, S.; Hruby, V. J. HPLC of peptides at lowered temperatures. <None Specified> . 1991. Tessek application note No.64. 1783 1991Tessek.pdf

  172. Lebl, M.; Stierandova, A.; Eichler, J.; Bienert, M. Alternative carriers and methods in solid phase synthesis. In: Peptides 90, Proc.21.EPS, Giralt, E., Andreu, D., Eds.; ESCOM: Leiden, 1991; pp 153-155. 1991Proc21EPS_153.pdf

  173. Lebl, M.; Fang, S.; Hruby, V. J. High-performance liquid chromatography of peptides at reduced temperatures: Separation of isomers. J. Chromatogr. 1991, 586 (1), 145-148. 1991JChromatogr.pdf

  174. Malat, J.; Lebl, M.; Ubik, K. Collision-induced liquid secondary ion mass spectra of oxytocin derivatives. A study of the influence of modifications in the disulfide bond on the adjacent peptide bond cleavage. Rapid Commun. Mass Spectrom. 1991, 5 (7), 316-318. 1991RapidCommMassSpec.pdf

  175. Patek, M.; Lebl, M. Safety-catch anchoring linkage for synthesis of peptide amides by Boc/Fmoc strategy. Tetrahedron Lett. 1991, 32, 3891-3894. 1991TetLett.pdf

  176. Prochazka, Z.; Zertova, M.; Barth, T.; Slaninova, J.; Maletinska, L.; Blaha, I.; Lebl, M. Vasopressin analogs as strong uterotonic inhibitors. In: Peptides 90, Proc.21.EPS, Giralt, E., Andreu, D., Eds.; ESCOM: Leiden, 1991; pp 663-664. 1991Proc21EPS_663.pdf

  177. Sepetov, N. F.; Lebl, M.; Krymsky, M. Sequence inversion and racemization of peptides containing glycine in position 3. In: Peptides 90, Proc.21.EPS, Giralt, E., Andreu, D., Eds.; ESCOM: Leiden, 1991; pp 84-85. 1991Proc21EPS_084.pdf

  178. Sepetov, N. F.; Krymsky, M. A.; Ovchinnikov, M. V.; Bespalova, Z. D.; Isakova, O. L.; Soucek, M.; Lebl, M. Rearrangement, racemization and decomposition of peptides in aqueous solution. Peptide Res. 1991, 4 (5), 308-313. 1991PeptRes_309.pdf

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  180. Eichler, J.; Bienert, M.; Sepetov, N. F.; Stolba, P.; Krchnak, V.; Smekal, O.; Gut, V.; Lebl, M. Cotton-carrier for solid phase peptide synthesis. In: Innovations and Perspectives in Solid Phase Synthesis, Epton, R., Ed.; SPCC: Birmingham, 1990; pp 337-343. 1990InnovPerspSPS_337.pdf

  181. Lebl, M.; Hill, P.; Kazmierski, W.; Karaszova, L.; Slaninova, J.; Fric, I.; Hruby, V. J. Conformationally restricted analogs of oxytocin; stabilization of inhibitory conformation. Int. J. Peptide Prot. Res. 1990, 36 (4), 321-330. 1990IntJPeptProtRes_321.pdf

  182. Lebl, M.; Gut, V.; Eichler, J. Continuous solid-phase synthesis. In: Peptides: Chemistry, Structure and Biology,Proc.11.APS, Rivier, J. E., Marshall, G. R., Eds.; ESCOM: Leiden, 1990; pp 1059-1060. 1990Proc11APS_1059.pdf

  183. Malat, J.; Ubik, K.; Lebl, M. Daughter ion mass spectra of oxytocin derivatives with modified disulfide bonds. Les Cahiers de Spectra 2000 1990, Suppl. 150, 54. 1990LeCahSpec.pdf

  184. Patek, M.; Lebl, M. A safety-catch type of amide protecting group. Tetrahedron Lett. 1990, 31, 5209-5212. 1990TetLett.pdf

  185. Prochazka, Z.; Ancans, J. E.; Slaninova, J.; Machova, A.; Barth, T.; Lebl, M. Synthesis and biological properties of vasopressin analogues containing 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid. Collect. Czech. Chem. Commun. 1990, 55, 1099-1105. 1990CCCC_1099.pdf

  186. Slaninova, J.; Barth, T.; Lebl, M.; Cerny, B.; Trojnar, J. Bioavailability of carbetocin ([2-O-methyltyrosine]deamino-1-carba-oxytocin) in the rat. In: Peptides: Chemistry, Structure and Biology,Proc.11.APS, Rivier, J. E., Marshall, G. R., Eds.; ESCOM: Leiden, 1990; pp 297-298. 1990Proc11APS_297.pdf

  187. Toth, G.; Lebl, M.; Hruby, V. J. Chiral thin-layer chromatographic separation of phenylalanine and tyrosine derivatives. J. Chromatogr. 1990, 504, 450-455. 1990JChromatogr.pdf

  188. Zertova, M.; Prochazka, Z.; Blaha, I.; Barth, T.; Slaninova, J.; Lebl, M. The analogues of 8-D-homoarginine-vasopressin with modification in position 2; Synthesis and some biological properties. Collect. Czech. Chem. Commun. 1990, 55, 3000-3007. 1990CCCC_3000.pdf

  189. Castrucci, A. M. L.; Lebl, M.; Hruby, V. J.; Matsunaga, T. O.; Hadley, M. E. Melanin concentrating hormone (MCH): The message sequence. Life Sci. 1989, 45 (13), 1141-1148. 1989LifeSci_1141.pdf

  190. Castrucci, A. M. L.; Hadley, M. E.; Lebl, M.; Zechel, C.; Hruby, V. J. Melanocyte stimulating hormone and melanin concentrating hormone may be structurally and evolutionarily related. Regul. Peptides 1989, 24 (1), 27-35. 1989RegPeptides.pdf

  191. Eichler, J.; Beyermann, M.; Bienert, M.; Lebl, M. Simultaneous peptide synthesis using cellulose paper as support material. In: Peptides 1988,Proc.20.EPS, Jung, G., Bayer, E., Eds.; Walter de Gruyter & Co.: Berlin, 1989; pp 205-207. 1989Proc20EPS_205.pdf

  192. Krchnak, V.; Vagner, J.; Eichler, J.; Lebl, M. Color monitored solid phase peptide synthesis. In: Peptides 1988,Proc.20.EPS, Jung, G., Bayer, E., Eds.; Walter de Gruyter & Co.: Berlin, 1989; pp 232-234. 1989Proc20EPS_232.pdf

  193. Lebl, M.; Barth, T.; Slaninova, J.; Hrbas, P.; Eichler, J.; Cerny, B. Synthesis, tritiation and biological studies with [2-O-methyltyrosine, 7-(3,4-dehydroproline)]deamino-1-carba-oxytocin. In: Peptides 1988,Proc.20.EPS, Jung, G., Bayer, E., Eds.; Walter de Gruyter & Co.: Berlin, 1989; pp 546-548. 1989Proc20EPS_546.pdf

  194. Lebl, M.; Slaninova, J.; Johnson, R. L. Analogs of oxytocin containing a pseudopeptide Leu-Gly bond of cis and trans configuration. Int. J. Peptide Prot. Res. 1989, 33, 16-21. 1989IntJPeptProtRes_16.pdf

  195. Lebl, M.; Hruby, V. J.; Castrucci, A. M. L.; Hadley, M. E. Melanin concentrating hormone analogues: Contraction of the cyclic structure. II.Antagonist activity. Life Sci. 1989, 44 (7), 451-457. 1989LifeSci_0451.pdf

  196. Lebl, M.; Eichler, J. Simulation of continuous solid phase synthesis: Synthesis of methionine enkephalin and its analogs. Peptide Res. 1989, 2 (4), 297-300. 1989PeptRes_297.pdf

  197. Matsunaga, T. O.; Hruby, V. J.; Lebl, M.; Castrucci, A. M. L.; Hadley, M. E. Melanin concentrating hormone (MCH): Structure-function aspects of its melanocyte stimulating hormone-like (MSH-like) activity. Peptides 1989, 10, 773-778. 1989Peptides.pdf

  198. Slaninova, J.; Lebl, M.; Eichler, J. Synthesis and properties of antiparallel dimer of deamino-1-carba-oxytocin. In: Peptides 1988,Proc.20.EPS, Jung, G., Bayer, E., Eds.; Walter de Gruyter & Co.: Berlin, 1989; pp 543-545. 1989Proc20EPS_543.pdf

  199. Zicha, J.; Kunes, J.; Lebl, M.; Pohlova, I.; Slaninova, J.; Jelinek, J. Antidiuretic and pressor actions of vasopressin in age-dependent DOCA-salt hypertension. Amer. J. Physiol. 1989, 256 (1;Part 2), R138-R145. 1989AmJPhysiol.pdf

  200. Bendlova, B.; Lebl, M.; Stolba, P.; Starka, L. Synthesis of modified human C-peptide and its fragments. Collect. Czech. Chem. Commun. 1988, 53, 2637-2644. 1988CCCC_2637.pdf

  201. Fassina, G.; Lebl, M.; Chaiken, I. Screening the recognition properties of peptide hormone sequence mutants by analytical high performance liquid affinity chromatography on immobilized neurophysin. Collect. Czech. Chem. Commun. 1988, 53, 2627-2636. 1988CCCC_2627.pdf

  202. Krchnak, V.; Vagner, J.; Safar, P.; Lebl, M. Noninvasive continuous monitoring of solid phase peptide synthesis by acid-base indicator. Collect. Czech. Chem. Commun. 1988, 53, 2542-2548. 1988CCCC_2542.pdf

  203. Krchnak, V.; Vagner, J.; Lebl, M. Noninvasive continuous monitoring of solid phase peptide synthesis by acid-base indicator (preliminary communication). Int. J. Peptide Prot. Res. 1988, 32 (5), 415-416. 1988IntJPeptProtRes_415.pdf

  204. Lebl, M.; Hruby, V. J.; Castrucci, A. M. L.; Visconti, M. A.; Hadley, M. E. Melanin concentrating hormone analogues: Contraction of the cyclic structure. 1.Agonist activity. J. Med. Chem. 1988, 31 (5), 949-954. 1988JMedChem.pdf

  205. Mader, P.; Vesela, V.; Heyrovsky, M.; Lebl, M.; Braunsteinova, M. Polarography of the oxytocin and vasopressin synthetic analogs. Collect. Czech. Chem. Commun. 1988, 53, 1579-1605. 1988CCCC_1579.pdf

  206. Prochazka, Z.; Ancans, J. E.; Slaninova, J.; Machova, A.; Barth, T.; Skopkova, J.; Budesinsky, M.; Pavlikova, F.; Lebl, M. Synthesis and properties of analogues of vasopressin with 1-aminocyclopropane-1-carboxylic acid. Collect. Czech. Chem. Commun. 1988, 53, 2604-2616. 1988CCCC_2604.pdf

  207. Barth, T.; Slaninova, J.; Lebl, M.; Hruby, V. J. Effect of threonine in position 4 in oxytocin and vasotocin analogs on the time course of uterotonic response. Endocrinol. Exper. 1987, 21 (3), 191-197. 1987EndocrinolExper.pdf

  208. Hruby, V. J.; Lebl, M. Conformational properties of neurohypophyseal hormone analogs in solution as determined by NMR and laser Raman spectroscopies. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 105-155.

  209. Jost, K.; Lebl, M.; Brtnik, F. Nomenclature. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 5-8.

  210. Jost, K.; Lebl, M.; Brtnik, F. Introductory remarks. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 1-4.

  211. Lebl, M. Analogs with dissociated and/or high activities. II.Uterotonic activity. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 78-102.

  212. Lebl, M.; Jost, K.; Brtnik, F. Tables of analogs. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 127-268.

  213. Lebl, M.; Sugg, E. E.; Van Binst, G.; van der Elst, P.; Tourwe, D.; Slaninova, J.; Hruby, V. J. Analogs of oxytocin containing a modified peptide bond. Int. J. Peptide Prot. Res. 1987, 30 (3), 318-322. 1987IntJPeptProtRes_318.pdf

  214. Lebl, M. Analogs with dissociated and/or high activities. III. Galactogogic activity. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 102-109.

  215. Lebl, M. Analogs with dissociated and/or high activities. I.Introduction. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 75-78.

  216. Lebl, M. Synthesis, purification, and stability of the neurohypophyseal hormone analogs. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 23-82.

  217. Lebl, M. Modification of other functional groups. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 156-160.

  218. Lebl, M. Isotopically modified analogs. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 83-104.

  219. Lebl, M.; Sugg, E. E.; Hruby, V. J. Proton NMR spectroscopic evidence for sulfur-aromatic interactions in peptides. Int. J. Peptide Prot. Res. 1987, 29 (1), 40-45. 1987IntJPeptProtRes_040.pdf

  220. Lebl, M. Analogs with inhibitory properties. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 17-74.

  221. Lebl, M.; Hruby, V. J. Other methods used in the investigation of neurohypophyseal hormone analog conformations. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 155-159.

  222. Lebl, M.; Fric, I.; Sugg, E. E.; Cody, W. L.; Hruby, V. J. Conformational studies of carba-analogs of oxytocin. In: Peptides 1986, Proc.19.EPS, Theodoropoulos, D., Ed.; Walter de Gruyter & Co.: Berlin, 1987; pp 341-344. 1986Proc19EPS_341.pdf

  223. Zaoral, M.; Blaha, I.; Lebl, M.; Barth, T. Vasopressin analogs with strong agonistic-antagonistic properties. In: Peptides 1986, Proc.19.EPS, Theodoropoulos, D., Ed.; Walter de Gruyter & Co.: Berlin, 1987; pp 465-468. 1986Proc19EPS_465.pdf

  224. Zicha, J.; Kunes, J.; Lebl, M.; Pohlova, I.; Jelinek, J. Haemodynamics and the participation of pressor systems in young and adult rats with age-dependent doca-salt hypertension. Physiol. Bohemoslov. 1987, 36, 89-92. 1987PhysiolBohem.pdf

  225. Hermann, P.; Jannasch, R.; Lebl, M. Application of high-performance liquid chromatography and capillary isotachophoresis to the purification and characterization of products of peptide synthesis. J. Chromatogr. 1986, 351, 283-293. 1986JChromatogr.pdf

  226. Hrbas, P.; Barth, T.; Lebl, M.; Papsuevich, A. O.; Flegel, M. Mono- and diiodo-derivatives of neurohypophysial hormones and their analogues. Beitr. Wirkstofforsch. 1985, 24, 182-187. 1985BeitrWirkst.pdf

  227. Lebl, M.; Drasar, P.; Koroniak, H.; Milecki, J.; Ikonomov, O. C. Nejnovejsí poznatky v chemii porkanovych sloucenin. Chem. Listy 1985, 79, 410-417. 1985ChemListy.pdf

  228. Lebl, M. Carba analogues of neurohypophysial hormones. In: Handbook of the Use of High Performance Liquid Chromatography for the Analytical and Preparative Separation of Amino Acids, Peptides and Proteins, Hancock, W. S., Ed.; CRC Press: Boca Raton, 1985; pp 169-178. 1985HandbookHPLC.pdf

  229. Lebl, M.; Barth, T.; Servitova, L.; Slaninova, J.; Jost, K. Oxytocin analogues with inhibitory properties, containing in position 2 a hydrophobic amino acid of D-configuration. Collect. Czech. Chem. Commun. 1985, 50, 132-145. 1985CCCC_0132.pdf

  230. Lebl, M.; Hruby, V. J.; Slaninova, J.; Barth, T. Solid phase synthesis and biological activities of oxytocin carba analogues containing threonine in position 4. Collect. Czech. Chem. Commun. 1985, 50, 418-427. 1985CCCC_0418.pdf

  231. Hrbas, P.; Skopkova, J.; Zicha, J.; Barth, T.; Lebl, M.; Jost, K. Nacartocin - analogue of oxytocin with enhanced natriuretic properties: natriuretic and hemodynamic characteristics. Endocrinol. Exper. 1984, 18 (2), 117-124. 1984EndocrinolExper.pdf

  232. Lebl, M.; Cody, W. L.; Wilkes, B. C.; Hruby, V. J.; Castrucci, A. M. L.; Hadley, M. E. Modification of the disulfide bridge in cyclic melanotropins. Collect. Czech. Chem. Commun. 1984, 49, 2680-2688. 1984CCCC_2680.pdf

  233. Lebl, M.; Cody, W. L.; Hruby, V. J. Cyclic melanotropins. Part VI. Reverse phase HPLC studies. J. Liq. Chromatogr. 1984, 7, 1195-1210. 1984JLiqChrom.pdf

  234. Lebl, M.; Barth, T.; Crankshaw, D. J.; Cerny, B.; Daniel, E. E.; Grover, A. K.; Jost, K. Synthesis and properties of [2-[3,5-(3)H2]-tyrosine,4-glutamic acid]deamino-1-carba-oxytocin. Collect. Czech. Chem. Commun. 1984, 49, 1921-1926. 1984CCCC_1921.pdf

  235. Lebl, M.; Hruby, V. J. Synthesis of cyclic peptides by solid phase technology. Tetrahedron Lett. 1984, 25 (20), 2067-2068. TetLett1984.pdf

  236. Lebl, M.; Barth, T.; Servitova, L.; Slaninova, J.; Hrbas, P. Synthesis and properties of carba-6-analogues of oxytocin containing a deaminopenicillamine residue in position 1. Collect. Czech. Chem. Commun. 1984, 49, 2012-2023. 1984CCCC_2012.pdf

  237. Lebl, M.; Cody, W. L.; Wilkes, B. C.; Hruby, V. J.; Castrucci, A. M. L.; Hadley, M. E. Cyclic melanotropins. Part VII: Modified ring structures: Synthesis and biological activity. Int. J. Peptide Prot. Res. 1984, 24 (5), 472-479. 1984IntJPeptProtRes_472.pdf

  238. Prochazka, Z.; Lebl, M.; Barth, T.; Hlavacek, J.; Trka, A.; Budesinsky, M.; Jost, K. Synthesis and properties of oxytocin analogues modified in the tripeptide side chain. Collect. Czech. Chem. Commun. 1984, 49, 642-652. 1984CCCC_0642.pdf

  239. Skopkova, J.; Barth, T.; Hrbas, P.; Jost, K.; Lebl, M. Natriuretic properties of [2-p-ethylphenylalanine]deamino-6- carba-oxytocin (Nacartocin) in cats. Exp. Clin. Endocrinol. 1984, 84, 235-238. 1984ExpClinEndocrinol.pdf

  240. Barth, T.; Lebl, M.; Jost, K.; Cantau, B.; Butlan, D.; Guillon, G.; Jard, S. Interactions of deamino-6-carba-oxytocin analogues in rat kidney and liver membrane systems. In: Peptides 1982,Proc.17.EPS, Blaha, K., Malon, P., Eds.; Walter de Gruyter: Berlin, 1983; pp 467-470. 1983Proc17EPS_467.pdf

  241. Barth, T.; Cantau, B.; Butlen, D.; Guillon, G.; Jard, S.; Lebl, M.; Jost, K. Oxytocin and vasopressin analogues capable of competition with vasopressin binding to rat liver membranes. Collect. Czech. Chem. Commun. 1983, 48, 1788-1795. 1983CCCC_1788.pdf

  242. Budesinsky, M.; Jezek, J.; Krchnak, V.; Lebl, M.; Zaoral, M.; Rotta, J.; Straka, R. Synthetic fragments of bacterial cell walls. Physicochemical and biological properties. In: Peptides 1982,Proc.17.EPS, Blaha, K., Malon, P., Eds.; Walter de Gruyter: Berlin, 1983; pp 305-310. 1983Proc17EPS_305.pdf

  243. Butlen, D.; Barth, T.; Cantau, B.; Guillon, G.; Jard, S.; Lebl, M.; Brtnik, F.; Jost, K. The structural requirements of oxytocin and vasopressin analogues for the activation of adenylate cyclase in the rat kidney medullary membrane system. Collect. Czech. Chem. Commun. 1983, 48, 3166-3176. 1983CCCC_3166.pdf

  244. Krojidlo, M.; Flegel, M.; Lebl, M. Method for cyclization of carba analogues of oxytocin. In: Peptides 1982,Proc.17.EPS, Blaha, K., Malon, P., Eds.; Walter de Gruyter: Berlin, 1983; pp 199-202. 1983Proc17EPS_199.pdf

  245. Lebl, M.; Barth, T.; Servitova, L.; Slaninova, J.; Jost, K. Analogues of neurohypophysial hormones containing a D-amino acid in position 2. In: Peptides 1982,Proc.17.EPS, Blaha, K., Malon, P., Eds.; Walter de Gruyter: Berlin, 1983; pp 457-460. 1983Proc17EPS_457.pdf

  246. Lebl, M. Analogues of neurohypophysial hormones with inhibitory effect on the pressoric activity of vasopressin. In: Vasopressin and Pathology of the Cardiovascular System in Aging, Chebotarev, D. F., Frolkis, V. V., Eds.; Institute of Gerontology: Kiev, 1983; pp 108-114. 1983VasopPathCardioSystAging.pdf

  247. Lebl, M.; Barth, T. Synthesis and some activities of [1-penicillamine]deamino-6-carba-oxytocin. In: Peptides:Structure and Function,Proc.8.APS, Hruby, V. J., Rich, D. H., Eds.; Pierce: Rockford, 1983; pp 357-360. 1983Proc8APS_357.pdf

  248. Lebl, M.; Gut, V. Calculation of the rate constant of a reversible reaction from the chromatographic peaks for muranyl dipeptide anomers. J. Chromatogr. 1983, 260, 478-482. JChromatogr1983_Gut.pdf

  249. Lebl, M. Amino acids and peptides CLXXXI. Separation of diastereoisomers of oxytocin analogues. J. Chromatogr. 1983, 264, 459-462. 1983JChromatogr_459.pdf

  250. Prochazka, Z.; Lebl, M.; Barth, T.; Hlavacek, J.; Jost, K. Two analogues of oxytocin with modified proline cyclic structure. In: Peptides 1982,Proc.17.EPS, Blaha, K., Malon, P., Eds.; Walter de Gruyter: Berlin, 1983; pp 441-444. 1983Proc17EPS_441.pdf

  251. Lebl, M.; Pospisek, J.; Hlavacek, J.; Barth, T.; Malon, P.; Servitova, L.; Hauzer, K.; Jost, K. Analogues of neurohypophysial hormones containing tert.leucine: synthesis and properties. Collect. Czech. Chem. Commun. 1982, 47, 689-701. 1982CCCC_0689.pdf

  252. Lebl, M. Correlation between hydrophobicity of substituents in the phenylalanine moiety of oxytocin carba-analogues and reversed- phase-chromatographic k' values. J. Chromatogr. 1982, 242, 342-345. 1982JChromatogr.pdf

  253. Lebl, M.; Hrbas, P.; Skopkova, J.; Slaninova, J.; Machova, A.; Barth, T.; Jost, K. Synthesis and properties of oxytocin analogues with high and selective natriuretic activity. Collect. Czech. Chem. Commun. 1982, 47, 2540-2560. 1982CCCC_2540.pdf

  254. Barth, T.; Hrbas, P.; Skopkova, J.; Slaninova, J.; Lebl, M.; Jost, K. Natriuretic effects of oxytocin analogues. In: Peptides 1980,Proc.16.EPS, Brunfeldt, K., Ed.; Scriptor: Copenhagen, 1981; pp 416-419. 1981Proc16EPS_416.pdf

  255. Barth, T.; Slaninova, J.; Servitova, L.; Lebl, M.; Kotsira-Engonopoulos, C.; Tzougraki, C.; Photaki, I.; Krojidlo, M.; Jost, K. The effect of some structural modification of the oxytocin molecule on the duration of the galactogogic response. Collect. Czech. Chem. Commun. 1981, 46, 2441-2445. 1981CCCC_2441.pdf

  256. Bienert, M.; Lebl, M.; Mehlis, B.; Niedrich, H. Synthesis and application of methionin S-tert-butylsulfonium peptides. In: Peptides 1980,Proc.16.EPS, Brunfeldt, K., Ed.; Scriptor: Copenhagen, 1981; pp 127-132. 1981Proc16EPS_127.pdf

  257. Lebl, M.; Barth, T.; Jost, K. Chromatographic and pharmacological properties of carba- analogues of neurohypophyseal hormones sulfoxides. A general method of sulfoxide group determination in peptides. In: Peptides 1980,Proc.16.EPS, Brunfeldt, K., Ed.; Scriptor: Copenhagen, 1981; pp 719-724. 1981Proc16EPS_719.pdf

  258. Prochazka, Z.; Lebl, M.; Servitova, L.; Barth, T.; Jost, K. Synthesis and pharmacological properties of 2-p-fluorophenyl- alanine deamino-1-carba-oxytocin and of its diastereoisomeric sulfoxides. Collect. Czech. Chem. Commun. 1981, 46, 947-956. 1981CCCC_0947.pdf

  259. Slaninova, J.; Lebl, M.; Barth, T.; Jost, K. The effect of magnesium ions on the uterotonic activity of carba analogues of oxytocin modified in position 4. Collect. Czech. Chem. Commun. 1981, 46, 1689-1692. 1981CCCC_1689.pdf

  260. Barth, T.; Slaninova, J.; Lebl, M.; Jost, K. Biological activities and protracted action of carba-analogues of deamino-oxytocin with O-methyltyrosine in position 2. Collect. Czech. Chem. Commun. 1980, 45, 3045-3050. 1980CCCC_3045.pdf

  261. Hrbas, P.; Barth, T.; Skopkova, J.; Lebl, M.; Jost, K. Effect of some oxytocin analogues on natriuresis in rats. Endocrinol. Exper. 1980, 14 (2), 151-157. 1980EndocrinolExper.pdf

  262. Hrbas, P.; Skopkova, J.; Barth, T.; Lebl, M.; Jost, K. Renal sodium excretion in rats. Effect of amino acid replacement in position 4 of the oxytocin molecule. In: Hormonal Regulation of Sodium Excretion, Lichardus, B., Schrier, R. W., Ponec, J., Eds.; Elsevier: Amsterdam, 1980; pp 169-172. 1980HormRegSodExcr_169.pdf

  263. Lebl, M. High-performance liquid chromatography of carba analogues of oxytocin; a method for the determination of sulfides and sulfoxides in peptides. Collect. Czech. Chem. Commun. 1980, 45, 2927-2937. 1980CCCC_2927.pdf

  264. Lebl, M.; Machova, A.; Hrbas, P.; Barth, T.; Jost, K. Analogues of deamino-1-carba-oxytocin with aliphatic amino acid in position 4: Chemical synthesis and biological activities. Collect. Czech. Chem. Commun. 1980, 45, 2714-2723. 1980CCCC_2714.pdf

  265. Lebl, M.; Barth, T.; Skopkova, J.; Jost, K. Synthesis and some pharmacological properties of [7-glycine,8- ornithine]-vasopressin and of its two analogues. Collect. Czech. Chem. Commun. 1980, 45, 2865-2871. 1980CCCC_2865.pdf

  266. Lebl, M.; Barth, T.; Jost, K. Synthesis and pharmacological properties of oxytocin analogues modified simultaneously in position 2 and in the disulfide bridge. Collect. Czech. Chem. Commun. 1980, 45, 2855-2864. 1980CCCC_2855.pdf

  267. Skopkova, J.; Hrbas, P.; Barth, T.; Lebl, M.; Jost, K. Renal sodium excretion in rats. Effect of structural modification of position 2 of deamino-6-carba-oxytocin. In: Hormonal Regulation of Sodium Secretion, Lichardus, B., Schrier, R. W., Ponec, J., Eds.; Elsevier: Amsterdam, 1980; pp 163-168. 1980HormRegSodExcr_163.pdf

  268. Barth, T.; Lebl, M.; Bojanovska, V.; Jost, K. Analogues of oxytocin acting as irreversible inhibitors of oxytocin. In: Peptides 1978,Proc.15.EPS, Siemion, I. Z., Kupryszewski, G., Eds.; Wroclaw University Press: Wroclaw, 1979; pp 475-479. 1979Proc15EPS_475.pdf

  269. Lebl, M.; Dimeli, A.; Bojanovska, V.; Slaninova, J.; Barth, T.; Jost, K. Synthesis and some biological properties of amides derived from [4-glutamic acid]deamino-1-carba-oxytocin. Collect. Czech. Chem. Commun. 1979, 44, 2556-2562. 1979CCCC_2556.pdf

  270. Lebl, M.; Bojanovska, V.; Barth, T.; Jost, K. Synthesis and properties of oxytocin analogues acting as irreversible inhibitors of the uterotonic response to oxytocin. Collect. Czech. Chem. Commun. 1979, 44, 2573-2582. 1979CCCC_2573.pdf

  271. Lebl, M.; Barth, T.; Jost, K. Analogues of oxytocin with esters of glutamic acid instead of glutamine in position 4: synthesis of a compound with high and specific galactogogic activity. Collect. Czech. Chem. Commun. 1979, 44, 2563-2572. 1979CCCC_2563.pdf

  272. Lebl, M.; Jost, K. Selective oxidation of sulfur in peptide synthesis. In: Peptides 1978,Proc.15.EPS, Siemion, I. Z., Kupryszewski, G., Eds.; Wroclaw University Press: Wroclaw, 1979; pp 109-112. 1979Proc15EPS_109.pdf

  273. Lebl, M.; Barth, T.; Jost, K. Synthesis, reduction, and pharmacological properties of the sulfoxides of some carba-analogues of oxytocin. Collect. Czech. Chem. Commun. 1978, 43, 1538-1556. 1978CCCC_1538.pdf

  274. Lebl, M.; Jost, K. Mechanismus racemisace derivátu aminokyselin. Chem. Listy 1978, 72, 252-266. 1978ChemListy.pdf

  275. Lebl, M.; Jost, K. Synthesis of [4-glutamic acid]deamino-1-carba-oxytocin. Collect. Czech. Chem. Commun. 1978, 43, 523-534. 1978CCCC_0523.pdf

  276. Lebl, M.; Barth, T.; Jost, K. Na-glycyl-glycyl-glycyl-8-ornithine-vasopressin: A trypsin resistant vasopressin analog with a specific pressor effect. Collect. Czech. Chem. Commun. 1978, 43, 1300-1305. 1978CCCC_1300.pdf

  277. Lebl, M.; Bojanovska, V.; Barth, T.; Jost, K. Oxytocin analogs effective as noncompetitive inhibitors in uterotonic test. Experientia 1978, 34 (12), 1543-1544. 1978Experientia.pdf

  278. Ferles, M.; Kocian, O.; Lebl, M.; Lovy, J.; Radl, S.; Silhankova, A.; Stern, P. Electrolytic reduction of quarternary salts of some alcohols of pyridine series, of corresponding alkylpyridines and alkenylpyridines. Collect. Czech. Chem. Commun. 1976, 41, 598-603. 1975CCCC_0598.pdf

  279. Ferles, M.; Lebl, M.; Silhankova, A.; Stern, P.; Wimmer, Z. Reduction of tertiary alcohols of the pyridine series and corresponding alkenylpyridines with zinc and formic acid. Collect. Czech. Chem. Commun. 1975, 40, 1571-1575. 1975CCCC_1571.pdf

  280. Ferles, M.; Lebl, M.; Stern, P.; Trska, P. Mixed electrolytic reduction of 1,4,-dimethylpyridinium methylsulfate with acetone and of 1-methylpyridinium methylsulfate with cyclopentanone. Collect. Czech. Chem. Commun. 1975, 40, 2183-2190. 1975CCCC_2183.pdf