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PAPERS PUBLISHED

  1. Kozlov,I.A., Melnyk,P.C., Hachmann,J.P., Srinivasan,A., Shults,M.D., Zhao,C., Musmacker,J., Nelson,N., Barker,D.L., & Lebl,M. (2008) A high-complexity, multiplexed solution-phase assay for profiling protease activity on microarrays. Comb. Chem. High Throughput Screening, 11, 24-35. #20880 (Available on Internet)

  2. Kermani,B.G., Kozlov,I.A., Melnyk,P.C., Zhao,C., Hachmann,J.P., & Lebl,M. (2007) Using support vector machine regression to model the retention of peptides in immobilized metal-affinity chromatography. Sensors. and Actuators B: Chemical, 125, 149-157. #20821 (Available on Internet)

  3. Kozlov,I.A., Kermani,B.G., Melnyk,P.C., Barker,D.L., Zhao,C., Hachmann,J.P., & Lebl,M. (2007) Study of the retention of histidine containing peptides on nickel column. J. Chromatogr. Sci., 45, 207-211. #20817 (Available on Internet)

  4. Kozlov,I.A., Melnyk,P.C., Hachmann,J.P., Barker,D.L., Lebl,M., & Zhao,C. (2007) Evaluation of different chemical strategies for conjugation of oligonucleotides to peptides. Nucleosides, Nucleotides & Nucleic Acids, 26, 1353-1357. #20818 (Available on Internet)

  5. Lebl,M., Kozlov,I.A., Melnyk,P.C., Hachmann,J.P., Srinivasan,A., Shults,M.D., Musmacker,J., Nelson,N., Kermani,B.G., Zhao,C. & Barker,D.L. (2007) High complexity protease and kinase profiling solution assays with readout on randomly assembled microarrays. In Anonymous, Proc.29th Eur. Pept. Symp., Gdansk, 2006. (pp. in press. #20819 (Available on Internet)

  6. Raman,B., Kotseroglou,T., Clark,L., Lebl,M., & Gutierrez-Osuna,R. (2007) Neuromorphic processing for optical microbead arrays: dimensionality reduction and contrast enhancement. IEEE Sensors Journal, 7, 506-514. #20823 (Available on Internet)

  7. Shiryaev,S.A., Ratnikov,B.I., Aleshin,A.E., Kozlov,I.A., Nelson,N.A., Lebl,M., Smith,J.W., Liddington,R.C., & Strongin,A.Y. (2007) Switching the substrate specificity of the two-component NS2B-NS3 flaviviral proteinase by structure-based mutagenesis. J. Virol., 81, 4501-4509. #20879 (Available on Internet)

  8. Shiryaev,S.A., Kozlov,I.A., Ratnikov,B.I., Smith,J.W., Lebl,M., & Strongin,A.Y. (2007) Cleavage preference distinguishes the two-component NS2B-NS3 serine proteinases of Dengue and West Nile viruses. Biochem. J., 401, 743-752. #20820 (Available on Internet)

  9. Shults,M.D., Kozlov,I.A., Nelson,N., Kermani,B.G., Melnyk,P.C., Shevchenko,V., Srinivasan,A., Musmacker,J., Hachmann,J.P., Barker,D.L., Lebl,M., & Zhao,C. (2007) A Multiplexed Protein Kinase Assay. Chembiochem, 8, 933-942. #20822 (Available on Internet)

  10. Hachmann,J.P., & Lebl,M. (2006) Search for optimal coupling reagent in multiple peptide synthesizer. Biopolymers (Pept. Sci. ), 84, 340-347. #20815 (Available on Internet)

  11. Hachmann,J.P., & Lebl,M. (2006) Synthesis of poly d(G-C) oligonucleotides. Nucleosides, Nucleotides and Nucleic Acids, 25, 705-717. #20813 (Available on Internet)

  12. Hachmann,J.P., & Lebl,M. (2006) Alternative to piperidine in Fmoc solid phase synthesis. Journal of Combinatorial Chemistry, 8, 149. #20807 (Available on Internet)

  13. Kermani,B.G., Fomenko,I., Kotseroglou,T., Forood,B., Clark,L., Barker,D., & Lebl,M. (2006) Decoding beads in a randomly assembled optical nose. Sensors and Actuators B, 117, 282-285. #20814 (Available on Internet)

  14. Kozlov,I.A., Melnyk,P.C., Zhao,C., Hachmann,J.P., Shevchenko,V., Srinivasan,A., Barker,D.L., & Lebl,M. (2006) A method for rapid protease substrate evaluation and optimization. Comb. Chem. High Throughput Screening, 9, 481-487. #20816 (Available on Internet)

  15. Lebl,M. & Hachmann,J.P. (2005) High-throughput peptide synthesis. In J.Howl (Ed.), (pp. 167-194). Humana Press, Inc., Totowa, NJ. #20725 (Available on Internet)

  16. Lebl,M. (2005) Combinatorial Chemistry. In C.A.Hempstead & W.E.Worthington (Eds.), Encyclopedia of 20th-Century Technology. (pp. 171-174). Routledge, New York. #20726 (Available on Internet)

  17. Lebl,M., Pokorny,V., & Krchnak,V. (2005) Simple tools for resin distribution. Journal of Combinatorial Chemistry, 7, 42-45. #20722 (Available on Internet)

  18. Kermani,B., Fomenko,I., Kotseroglou,T., Forood,B., Clark,L., Barker,D. & Lebl,M. (2004) Supervised learning for decoding beads in a randomly-assembled optical nose. In Anonymous, Computational Biology Workshop, Neural Information Processing System (NIPS), 11th Annual Conference. Whistler, BC, Canada. #20729 (Available on Internet)

  19. Kermani,B., Kotseroglou,T., Forood,B., Barker,D. & Lebl,M. (2004) Optical nose signal denoising and detrending using wavelets. In Anonymous, Proceedings of 8th World Multiconference on Systems, Cybernetics, and Informatics. (pp. 148-149). Orlando, FL. #20728 (Available on Internet)

  20. Lebl,M. (2003) Centrifugation Based Automated Synthesis Technologies. J. Assoc. Lab. Autom., 8, 30-36. #18632 (Available on Internet)

  21. Forood,B., Kotseroglou,T., Clark,L., Lebl,M., Lieu,M.-H., Kermani,B., Barker,D. & Dickinson,T. (2002) Chemical detection using Illumina's BeadArray technology. In Anonymous, Proc. 9th International Symposium on Olfaction and Electronic Nose, ISOEN'02. Rome. #20727 (Available on Internet)

  22. Lam,K.S. & Lebl,M. (2002) Synthesis of One-Bead-One-Compound Combinatorial Peptide Library. In John M.Walker (Ed.), Protein Protocols on CD-ROM Version 2.0. (pp. 20-24). Humana Press, Totowa, NJ. #18633 (Available on Internet)

  23. Lebl, Michal Combinatorial chemistry: The history and the basics. In: Anonymous. (Eds.) Integrated Drug Discovery Technologies. #20394 (Available on Internet)

  24. Lebl, M. and Houghten, R. A. Preface. In: M.Lebl & R.A.Houghten. (Eds.) American Peptide Society, San Diego p.ix Peptides; The Wave of the Future. Proc. 2nd Int. 17th Amer. Pept. Symp. #20724 (Available on Internet)

  25. Lebl, M., Burger, C., Ellman, B., Heiner, D., Ibrahim, G., Jones, A., Nibbe, M., Pires, J., Mudra, P., Pokorny, V., Poncar, P., and Zenisek, K. Fully automated parallel oligonucleotide synthesizer. In: M.Lebl & R.A.Houghten. (Eds.) American Peptide Society, San Diego p.277 Peptides; The Wave of the Future. Proc. 2nd Int. 17th Amer. Pept. Symp. #18631 (Available on Internet)

  26. Lebl,M. & Pires,J. (2001) Solid-phase parallel synthesis of a large array of tetrahydroisoquinolinones. In I.Sucholeiki (Ed.), High-Throughput Synthesis. (pp. 197-205). Marcel Dekker, Inc., New York. #16464 (Available on Internet)

  27. Lebl,M., Pires,J., Burger,C., Ni,Y. & Chen,Y. (2001) Solid-phase parallel synthesis of large tetrahydroisoquinolinone library. In I.Sucholeiki (Ed.), High-Throughput Synthesis. (pp. 187-195). Marcel Dekker, Inc., New York. #16463 (Available on Internet)

  28. Lebl,M., Burger,C., Ellman,B., Heiner,D., Ibrahim,G., Jones,A., Nibbe,M., Thompson,J., Mudra,P., Pokorny,V., Poncar,P., & Zenisek,K. (2001) Fully automated parallel oligonucleotide synthesizer. Collect. Czech. Chem. Commun., 66, 1299-1314. #18630 (Available on Internet)

  29. Eichler,J., & Lebl,M. (2000) Combinatorial chemistry: A powerful tool for basic research and drug discovery. Journal of Clinical Ligand Assay, 23, 262-272. #16633 (Available on Internet)

  30. Lebl,M. (2000) New technique for high-throughput synthesis of peptides, peptidomimetics and nonpeptide small organic molecule arrrays. In G.B.Fields, J.P.Tam & G.Barany (Eds.), Peptides for the New Millennium. (pp. 164-166). Kluwer Academic Publisher, Dordrecht. #15715 (Available on Internet)

  31. Lebl,M., Ma,J., Pires,J., Dooley,C. & Houghten,R.A. (2000) Rapid parallel synthesis of 584 betides, peptides composed largely of beta-amino acids with side-chains not found in natural peptides. In G.B.Fields, J.P.Tam & G.Barany (Eds.), Peptides for the New Millennium. (pp. 174-175). Kluwer Academic Publisher, Dordrecht. #15719 (Available on Internet)

  32. Ni,Y., Krchnak,V., & Lebl,M. (2000) New approach for preparation of 2,3,7-trisubstituted 3,4-dihydroisoquinolinone libraries on solid phase. Mol. Diversity, 5, 153-161. #20494 (Available on Internet)

  33. Lebl,M. (1999) Parallel personal comments on "classical" papers in combinatorial chemistry. Journal of Combinatorial Chemistry, 1, 3-24. #12028 (Available on Internet)

  34. Lebl,M., Krchnak,V., Ibrahim,G., Pires,J., Burger,C., Ni,Y., Chen,Y., Podue,D., Mudra,P., Pokorny,V., Poncar,P., & Zenisek,K. (1999) Solid-phase synthesis of large tetrahydroisoquinolinone arrays by two different approaches. Synthesis-Stuttgart, 1971-1978. #13835 (Available on Internet)

  35. Lebl,M., Pires,J., Poncar,P., & Pokorny,V. (1999) Evaluation of gaseous hydrogen fluoride as a convenient reagent for parallel cleavage from the solid support. Journal of Combinatorial Chemistry, 1, 474-479. #13836 (Available on Internet)

  36. Lebl,M. (1999) Sooner or later someone else will cotton on to this idea (in " Matrix Assisted Synthetic Transformations: A Mosaic of Diverse Contributions. II. The Pattern Is Completed" by D. Hudson). Journal of Combinatorial Chemistry, 1, 438-442. #18636 (Available on Internet)

  37. Lebl,M. & Krchnak,V. (1999) Techniques for massively parallel synthesis of small organic molecules. In R.Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries. (pp. 43-46). Mayflower Scientific Limited, Birmingham. #10056 (Available on Internet)

  38. Lebl,M. (1999) Solid-phase synthesis of combinatorial libraries. Curr. Opin. Drug. Disc. Develop., 2, 385-395. #13357 (Available on Internet)

  39. Lebl, M. New approaches to automatic synthesis of large arrays of small organic molecules. In: Anonymous. (Eds.) Osaka, Japan p.6 Proceedings of combinatorial chemistry conference. #20723 (Available on Internet)

  40. Lebl,M. (1999) New technique for high-throughput synthesis. Bioorg. Med. Chem. Lett., 9, 1305-1310. #12856 (Available on Internet)

  41. Rinnova,M., Lebl,M., & Soucek,M. (1999) Solid-phase peptide synthesis by fragment condensation: Coupling in swelling volume. Lett. Peptide Sci., 6, 15-22. #13834 (Available on Internet)

  42. Rinnova,M., Soucek,M., Voburka,Z., Lebl,M. & Fusek,M. (1999) Sanger's reagent: An excellent end-capping and/or labeling agent for SPPS. In R.Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries. (pp. 385-386). Mayflower Scientific Limited, Birmingham. #13719 (Available on Internet)

  43. Thorpe,D.S., Yeoman,H., Chan,A.W.E., Krchnak,V., Lebl,M., & Felder,S. (1999) Combinatorial chemistry reveals a new motif that binds the platelet fibrinogen receptor, gpIIbIIIa. Biochem. Biophys. Res. Commun., 256, 537-541. #12667 (Available on Internet)

  44. Lam,K.S., & Lebl,M. (1998) Synthesis of a one-bead one-compound combinatorial peptide library. Methods in Molecular Biology (Totowa, New Jersey), 87, 1-6. #20693 (Available on Internet)

  45. Lebl,M. (1998) A new approach to automated solid phase synthesis based on centrifugation of tilted plates. J. Assoc. Lab. Autom., 3, 59-61. #11029 (Available on Internet)

  46. Lebl,M. (1998) Solid-phase synthesis on planar supports. Biopolymers (Pept. Sci. ), 47, 397-404. #12265 (Available on Internet)

  47. Ostrem,J.A., Al-Obeidi,F., Safar,P., Safarova,A., Stringer,S.K., Patek,M., Cross,M.T., Spoonamore,J., LoCascio,J.C., Kasireddy,P., Thorpe,D.S., Sepetov,N., Lebl,M., Wildgoose,P., & Strop,P. (1998) Discovery of a novel, potent, and specific family of factor Xa inhibitors via combinatorial chemistry. Biochemistry, 37, 1053-1059. #10581 (Available on Internet)

  48. Patek,M., & Lebl,M. (1998) Safety-catch and multiply cleavable linkers in solid-phase synthesis. Biopolymers (Pept. Sci. ), 47, 353-363. #12262 (Available on Internet)

  49. Seligmann,B., Lebl,M. & Lam,K.S. (1998) Solid-phase peptide synthesis, lead generation, and optimization. In E.M.Gordon & J.F.J.Kerwin (Eds.), Combinatorial Chemistry and Molecular Diversity in Drug Discovery. (pp. 39-109). John Wiley & Sons, New York. #11709 (Available on Internet)

  50. Cargill,J.F., & Lebl,M. (1997) New methods in combinatorial chemistry: Robotics and parallel synthesis. Curr. Opin. Chem. Biol., 1, 67-71. #8737 (Available on Internet)

  51. Krchnak,V., Weichsel,A.S., Lebl,M., & Felder,S. (1997) Automated solid-phase organic synthesis in micro-plate wells. Synthesis of N-(alkoxy-acyl)amino alcohols. Bioorg. Med. Chem. Lett., 7, 1013-1016. #6948 (Available on Internet) 4222

  52. Lam,K.S., Lebl,M., & Krchnak,V. (1997) The "one-bead one-compound" combinatorial library method. Chem. Rev., 97, 411-448. #6980 (Available on Internet) 4444

  53. Lebl,M., & Krchnak,V. (1997) Synthetic peptide libraries. Methods Enzymol., 289, 336-392. #9998 (Available on Internet)

  54. Chen,C.L., Strop,P., Lebl,M., & Lam,K.S. (1996) One bead-one compound combinatorial peptide library: Different types of screening. Methods Enzymol., 267, 211-219. #4785 (Available on Internet)

  55. Eichler,J., Houghten,R.A., & Lebl,M. (1996) Inclusion volume solid-phase peptide synthesis. J. Peptide Sci., 2, 240-244. #3547 (Available on Internet)

  56. Hruby,V.J., Shenderovich,M., Lam,K.S., & Lebl,M. (1996) Design considerations and computer modeling related to the development of molecular scaffolds and peptide mimetics for combinatorial chemistry. Mol. Diversity, 2, 46-56. #5324 (Available on Internet)

  57. Krchnak,V. & Lebl,M. (1996) MARS: Multiple automatic robot synthesizer featuring a novel timing procedure and random access to reagents and reaction vessels. In R.Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries. (pp. 93-96). Mayflower Scientific Limited, Birmingham. #6934 (Available on Internet) 3656

  58. Krchnak,V., Cabel,D., & Lebl,M. (1996) MARS: Multiple automated robotic synthesizer for continuous flow of peptides. Peptide Res., 9, 45-49. #3469 (Available on Internet)

  59. Krchnak,V., & Lebl,M. (1996) Synthetic library techniques: Subjective (biased and generic) thoughts and views. Mol. Diversity, 1, 193-216. #4806 (Available on Internet)

  60. Krchnak,V., Sepetov,N.F., Kocis,P., Patek,M., Lam,K.S. & Lebl,M. (1996) Combinatorial libraries of synthetic structures: Synthesis, screening, and structure determination. In R.Cortese (Ed.), Combinatorial Libraries: Synthesis, Screening and Application Potential. (pp. 27-52). Walter de Gruyter, Berlin. #2430 (Available on Internet)

  61. Krchnak,V., Weichsel,A.S., Cabel,D., Flegelova,Z., & Lebl,M. (1996) Structurally homogenous and heterogenous synthetic combinatorial libraries. Mol. Diversity, 1, 149-164. #4801 (Available on Internet)

  62. Krchnak,V., Weichsel,A.S., Cabel,D. & Lebl,M. (1996) Structurally homogenous and heterogenous libraries: Scaffold- based libraries and libraries built using bifunctional building blocks. In I.M.Chaiken & K.D.Janda (Eds.), Molecular Diversity and Combinatorial Chemistry. Libraries and Drug Discovery. (pp. 99-117). American Chemical Society, Washington,DC. #5101 (Available on Internet)

  63. Krchnak,V., Vagner,J., Flegelova,Z., Weichsel,A.S., Barany,G. & Lebl,M. (1996) Use of solid-phase Mitsunobu and Wittig reactions for contruction of peptide and non-peptide libraries. In P.T.P.Kaumaya & R.S.Hodges (Eds.), Peptides:Chemistry,Structure and Biology,Proc.14.APS. (pp. 307-308). Mayflower Scientific Ltd., Kingswinford. #3640 (Available on Internet)

  64. Lam,K.S. & Lebl,M. (1996) Combinatorial library based on the one-bead-one-compound concept. In G.Jung (Ed.), Combinatorial Peptide and Nonpeptide Libraries: A Handbook. (pp. 173-201). VCH, Weinheim. #2428 (Available on Internet)

  65. Lam,K.S., Lake,D., Salmon,S.E., Smith,J., Chen,M.L., Wade,S., Abdul-Latif,F., Leblova,Z., Ferguson,R.D., Krchnak,V., Sepetov,N.F., & Lebl,M. (1996) A one-bead one-peptide combinatorial library method for B-cell epitope mapping. Methods: A Companion to Methods in Enzymology, 9, 482-493. #5576 (Available on Internet)

  66. Lam,K.S., Lou,Q., Zhao,Z.G., Chen,M.L., Salmon,S.E., Wade,S. & Lebl,M. (1996) Identification and applications of idiotype-specific peptides for two murine B-cell lymphoma cell lines. In P.T.P.Kaumaya & R.S.Hodges (Eds.), Peptides:Chemistry,Structure and Biology,Proc.14.APS. (pp. 806-807). Mayflower Scientific Ltd., Kingswinford. #5066 (Available on Internet)

  67. Lebl,M., Krchnak,V., Strop,P. & Lam,K.S. (1996) Construction and screening of peptide and nonpeptide libraries based on one-bead-one-compound principle. In P.T.P.Kaumaya & R.S.Hodges (Eds.), Peptides:Chemistry,Structure and Biology,Proc.14.APS. (pp. 890-892). Mayflower Scientific Ltd., Kingswinford. #5057 (Available on Internet)

  68. Lebl,M., Krchnak,V., Patek,M., & Lam,K.S. (1996) Synthetic combinatorial libraries of scaffolded and unordered structures. Methods Mol. Cell. Biol., 6, 41-55. #7005 (Available on Internet) 3847

  69. Rinnova,M., Fusek,M. & Lebl,M. (1996) Use of methyl red in solid phase synthesis. In R.Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries. (pp. 509-510). Mayflower Scientific Limited, Birmingham. #3449 (Available on Internet)

  70. Rinnova,M., & Lebl,M. (1996) Molecular diversity and libraries of structures: Synthesis and screening. Collect. Czech. Chem. Commun., 61, 171-231. #3273 (Available on Internet)

  71. Salmon,S.E., Liu-Stevens,R.H., Zhao,Y., Lebl,M., Krchnak,V., Wertman,K., Sepetov,N., & Lam,K.S. (1996) High-volume cellular screening for anticancer agents with combinatorial chemical libraries: A new methodology. Mol. Diversity, 2, 57-63. #5331 (Available on Internet)

  72. Stankova,M., Strop,P., Chen,C. & Lebl,M. (1996) Mixtures of molecules versus mixtures of pure compounds on polymeric beads. In I.M.Chaiken & K.D.Janda (Eds.), Molecular Diversity and Combinatorial Chemistry. Libraries and Drug Discovery. (pp. 137-143). American Chemical Society, Washington,DC. #5103 (Available on Internet)

  73. Stankova,M., & Lebl,M. (1996) Library generation through successive substitution of trichlorotriazine. Mol. Diversity, 2, 75-80. #4844 (Available on Internet)

  74. Vagner,J., Barany,G., Lam,K.S., Krchnak,V., Sepetov,N.F., Ostrem,J.A., Strop,P., & Lebl,M. (1996) Enzyme-mediated spatial segregation on individual polymeric support beads: Application to generation and screening of encoded combinatorial libraries. Proc. Natl. Acad. Sci. USA, 93, 8194-8199. #147 (Available on Internet)

  75. Vagner,J., Krchnak,V., Lebl,M., & Barany,G. (1996) Solid-phase organic synthesis: Creation of carbon-carbon double bond under mild conditions by Wittig-type reactions. Collect. Czech. Chem. Commun., 61, 1697-1702. #7915 (Available on Internet)

  76. Flegelova,Z., Krchnak,V., Sepetov,N.F., Stankova,M., Issakova,O., Cabel,D., Lam,K.S. & Lebl,M. (1995) Libraries of small compact structures based on N-acyl-N-alkylamino acids. In H.L.S.Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 469-470). ESCOM, Leiden. #1347 (Available on Internet)

  77. Geysen,H.M., Houghten,R.A., Kauffman,S., Lebl,M., Moos,W.H., Pavia,M.R., & Szostak,J.W. (1995) Molecular diversity comes of age. Mol. Diversity, 1, 1-3. #8215 (Available on Internet)

  78. Kasal,A., Kohout,L., & Lebl,M. (1995) Synthesis of a scaffold for the creation of non-peptide libraries. Collect. Czech. Chem. Commun., 60, 2147-2155. #3467 (Available on Internet)

  79. Kocis,P., Issakova,O., Sepetov,N.F., & Lebl,M. (1995) Kemp's triacid scaffolding for synthesis of combinatorial nonpeptide uncoded libraries. Tetrahedron Lett., 36, 6623-6626. #3081 (Available on Internet)

  80. Krchnak,V., Flegelova,Z., Weichsel,A.S., & Lebl,M. (1995) Polymer-supported Mitsunobu ether formation and its use in combinatorial chemistry. Tetrahedron Lett., 36, 6193-6196. #2426 (Available on Internet)

  81. Krchnak,V., Weichsel,A.S., Issakova,O., Lam,K.S., & Lebl,M. (1995) Bifunctional scaffolds as templates for synthetic combinatorial libraries. Mol. Diversity, 1, 177-182. #4803 (Available on Internet)

  82. Krchnak,V., Weichsel,A.S., Cabel,D., & Lebl,M. (1995) Linear presentation of variable side-chain spacing in a highly diverse combinatorial library. Peptide Res., 8, 198-205. #2723 (Available on Internet)

  83. Lam,K.S., Wade,S., Abdul-Latif,F., & Lebl,M. (1995) Application of a dual color detection scheme in the screening of a random combinatorial peptide library. J. Immunol. Method, 180, 219-223. #2219 (Available on Internet)

  84. Lam,K.S. & Lebl,M. (1995) Peptide library screening based on the one-bead-one-peptide concept. In G.S.Lu, J.P.Tam & Y.C.Du (Eds.), Peptides:Biology and Chemistry,Proc.1994 Chinese Peptide Symposium. (pp. 273-277). ESCOM, Leiden. #2425 (Available on Internet)

  85. Lam,K.S., Lebl,M., Wu,J., Wade,S., Lou,Q., Zhao,Z.G., Chen,M.L., Chang,M.P., Smith,M. & Grimes,W.J. (1995) Peptide library screening based on the one-bead one-peptide concept: An update. In H.L.S.Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 453-454). ESCOM, Leiden. #1349 (Available on Internet)

  86. Lam,K.S., & Lebl,M. (1995) Synthesis and screening of a "one-bead-one-compound" combinatorial peptide library. Methods Mol. Cell. Biol., 6, 15-25. #8598 (Available on Internet)

  87. Lebl,M., Krchnak,V., Sepetov,N.F., Seligmann,B., Strop,P., Felder,S., & Lam,K.S. (1995) One-bead-one-structure combinatorial libraries. Biopolymers (Pept. Sci. ), 37, 177-198. #1782 (Available on Internet)

  88. Lebl,M., Krchnak,V., Sepetov,N.F., Nikolaev,V., Stankova,M., Kocis,P., Patek,M., Flegelova,Z., Ferguson,R. & Lam,K.S. (1995) Synthetic combinatorial libraries: A new tool for drug design. Methods for identifying the composition of compounds from peptide and/or nonpeptide libraries. In M.Z.Atassi & E.Appella (Eds.), Methods in Protein Structure Analysis. (pp. 335-342). Plenum Press, New York. #1353 (Available on Internet)

  89. Patek,M., Drake,B., & Lebl,M. (1995) Solid-phase synthesis of "small" organic molecules based on thiazolidine scaffold. Tetrahedron Lett., 36, 2227-2230. #1356 (Available on Internet)

  90. Safar,P., Stierandova,A. & Lebl,M. (1995) Amino-acid like subunits based on iminodiacetic acid and their application in linear and DKP libraries. In H.L.S.Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 471-472). ESCOM, Leiden. #1350 (Available on Internet)

  91. Salmon,S.E., Lam,K.S., Felder,S., Yeoman,H., Schlessinger,J., Ulrich,A., Krchnak,V., & Lebl,M. (1995) Use of large combinatorial chemical libraries for anticancer drug discovery. Int. J. Pharmacogn., 33 Suppl., 67-74. #5254 (Available on Internet)

  92. Seligmann,B., Abdul-Latif,F., Al-Obeidi,F., Flegelova,Z., Issakova,O., Kocis,P., Krchnak,V., Lam,K.S., Lebl,M., Ostrem,J., Safar,P., Sepetov,N., Stierandova,A., Strop,P., & Wildgoose,P. (1995) The construction and use of peptide and non-peptidic combinatorial libraries to discover enzyme inhibitors. Eur. J. Med. Chem., 30 (supplement); Pro, 319s-335s. #2429 (Available on Internet)

  93. Sepetov,N.F., Krchnak,V., Stankova,M., Lam,K.S., Wade,S. & Lebl,M. (1995) New approach in constructing and screening peptide libraries. In H.L.S.Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 467-468). ESCOM, Leiden. #1318 (Available on Internet)

  94. Sepetov,N.F., Krchnak,V., Stankova,M., Lam,K.S., Wade,S. & Lebl,M. (1995) Library of libraries: A novel approach in synthetic combinatorial libraries. In G.S.Lu, J.P.Tam & Y.C.Du (Eds.), Peptides:Biology and Chemistry,Proc.1994 Chinese Peptide Symposium. (pp. 271-272). ESCOM, Leiden. #3244 (Available on Internet)

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  100. Lam,K.S., Zhao,Z.G., Wade,S., Krchnak,V., & Lebl,M. (1994) Identification of small peptides that interact specifically with a small organic dye. Drug Develop. Res., 33, 157-160. #1009 (Available on Internet)

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  107. Madden,D., Krchnak,V., & Lebl,M. (1994) Synthetic combinatorial libraries: Views on techniques and their application. Perspect. Drug Disc. Design, 2, 269-286. #2431 (Available on Internet)

  108. Majer,P., Slaninova,J., & Lebl,M. (1994) Synthesis of methylated phenylalanines via hydrogenolysis of corresponding 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acids. Int. J. Peptide Prot. Res., 43, 62-68. #1638 (Available on Internet)

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  112. Prochazka,Z., Slaninova,J., Melin,P., Aurell,C.J., & Lebl,M. (1994) The deamino-carba analogs of vasotocin. Synthesis and some biological properties. Collect. Czech. Chem. Commun., 59, 421-428. #1288 (Available on Internet)

  113. Safar,P., Slaninova,J. & Lebl,M. (1994) The carba-modification of cystine-containing peptides: Synthesis of selectively protected cystathionines and their incorporation into the oxytocin molecule. In R.S.Hodges & J.A.Smith (Eds.), Peptides: Chemistry, Structure and Biology,Proc.13.APS. (pp. 119-120). ESCOM, Leiden. #1006 (Available on Internet)

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  117. Smith,M.H., Lam,K.S., Hersh,E.M., Lebl,M., & Grimes,W.J. (1994) Peptide sequences binding to MHC class I proteins. Mol. Immunol., 31, 1431-1437. #1007 (Available on Internet)

  118. Stankova,M., Wade,S., Lam,K.S., & Lebl,M. (1994) Synthesis of combinatorial libraries with only one representation of each structure. Peptide Res., 7, 292-298. #1754 (Available on Internet)

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  121. Vagner,J., Krchnak,V., Sepetov,N.F., Strop,P., Lam,K.S., Barany,G. & Lebl,M. (1994) Novel methodology for differentiation of "surface" and "interior" areas of poly(oxyethylene)-polystyrene (POE-PS) supports: Application to library screening procedures. In R.Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis. (pp. 347-352). Mayflower Worldwide Limited, Birmingham. #511 (Available on Internet)

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  180. Lebl,M., Slaninova,J., & Johnson,R.L. (1989) Analogs of oxytocin containing a pseudopeptide Leu-Gly bond of cis and trans configuration. Int. J. Peptide Prot. Res., 33, 16-21. #584 (Available on Internet)

  181. Lebl,M., Hruby,V.J., Castrucci,A.M.L., & Hadley,M.E. (1989) Melanin concentrating hormone analogues: Contraction of the cyclic structure. II.Antagonist activity. Life Sci., 44, 451-457. #1773 (Available on Internet)

  182. Lebl,M., Barth,T., Slaninova,J., Hrbas,P., Eichler,J. & Cerny,B. (1989) Synthesis, tritiation and biological studies with [2-O-methyltyrosine, 7-(3,4-dehydroproline)]deamino-1-carba-oxytocin. In G.Jung & E.Bayer (Eds.), Peptides 1988,Proc.20.EPS. (pp. 546-548). Walter de Gruyter & Co., Berlin. #1780 (Available on Internet)

  183. Lebl,M., & Eichler,J. (1989) Simulation of continuous solid phase synthesis: Synthesis of methionine enkephalin and its analogs. Peptide Res., 2, 297-300. #585 (Available on Internet)

  184. Matsunaga,T.O., Hruby,V.J., Lebl,M., Castrucci,A.M.L., & Hadley,M.E. (1989) Melanin concentrating hormone (MCH): Structure-function aspects of its melanocyte stimulating hormone-like (MSH-like) activity. Peptides, 10, 773-778. #1781 (Available on Internet)

  185. Slaninova,J., Lebl,M. & Eichler,J. (1989) Synthesis and properties of antiparallel dimer of deamino-1-carba-oxytocin. In G.Jung & E.Bayer (Eds.), Peptides 1988,Proc.20.EPS. (pp. 543-545). Walter de Gruyter & Co., Berlin. #1779 (Available on Internet)

  186. Zicha,J., Kunes,J., Lebl,M., Pohlova,I., Slaninova,J., & Jelinek,J. (1989) Antidiuretic and pressor actions of vasopressin in age-dependent DOCA-salt hypertension. Amer. J. Physiol., 256, R138-R145. #586 (Available on Internet)

  187. Bendlova,B., Lebl,M., Stolba,P., & Starka,L. (1988) Synthesis of modified human C-peptide and its fragments. Collect. Czech. Chem. Commun., 53, 2637-2644. #582 (Available on Internet)

  188. Fassina,G., Lebl,M., & Chaiken,I. (1988) Screening the recognition properties of peptide hormone sequence mutants by analytical high performance liquid affinity chromatography on immobilized neurophysin. Collect. Czech. Chem. Commun., 53, 2627-2636. #583 (Available on Internet)

  189. Krchnak,V., Vagner,J., & Lebl,M. (1988) Noninvasive continuous monitoring of solid phase peptide synthesis by acid-base indicator (preliminary communication). Int. J. Peptide Prot. Res., 32, 415-416. #1775 (Available on Internet)

  190. Krchnak,V., Vagner,J., Safar,P., & Lebl,M. (1988) Noninvasive continuous monitoring of solid phase peptide synthesis by acid-base indicator. Collect. Czech. Chem. Commun., 53, 2542-2548. #581 (Available on Internet)

  191. Lebl,M., Hruby,V.J., Castrucci,A.M.L., Visconti,M.A., & Hadley,M.E. (1988) Melanin concentrating hormone analogues: Contraction of the cyclic structure. 1.Agonist activity. J. Med. Chem., 31, 949-954. #1772 (Available on Internet)

  192. Mader,P., Vesela,V., Heyrovsky,M., Lebl,M., & Braunsteinova,M. (1988) Polarography of the oxytocin and vasopressin synthetic analogs. Collect. Czech. Chem. Commun., 53, 1579-1605. #580 (Available on Internet)

  193. Prochazka,Z., Ancans,J.E., Slaninova,J., Machova,A., Barth,T., Skopkova,J., Budesinsky,M., Pavlikova,F., & Lebl,M. (1988) Synthesis and properties of analogues of vasopressin with 1-aminocyclopropane-1-carboxylic acid. Collect. Czech. Chem. Commun., 53, 2604-2616. #1776 (Available on Internet)

  194. Barth,T., Slaninova,J., Lebl,M., & Hruby,V.J. (1987) Effect of threonine in position 4 in oxytocin and vasotocin analogs on the time course of uterotonic response. Endocrinol. Exper., 21, 191-197. #1768 (Available on Internet)

  195. Hruby,V.J. & Lebl,M. (1987) Conformational properties of neurohypophyseal hormone analogs in solution as determined by NMR and laser Raman spectroscopies. In K.Jost, M.Lebl & F.Brtnik (Eds.), CRC Handbook of Neurohypophyseal Hormone Analogs. (pp. 105-155). CRC Press, Boca Raton. #1660

  196. Jost,K., Lebl,M. & Brtnik,F. (1987) Introductory remarks. In K.Jost, M.Lebl & F.Brtnik (Eds.), CRC Handbook of Neurohypophyseal Hormone Analogs. (pp. 1-4). CRC Press, Boca Raton. #1656

  197. Jost,K., Lebl,M. & Brtnik,F. (1987) Nomenclature. In K.Jost, M.Lebl & F.Brtnik (Eds.), CRC Handbook of Neurohypophyseal Hormone Analogs. (pp. 5-8). CRC Press, Boca Raton. #1657

  198. Lebl,M., Sugg,E.E., & Hruby,V.J. (1987) Proton NMR spectroscopic evidence for sulfur-aromatic interactions in peptides. Int. J. Peptide Prot. Res., 29, 40-45. #1766 (Available on Internet)

  199. Lebl,M. (1987) Analogs with inhibitory properties. In K.Jost, M.Lebl & F.Brtnik (Eds.), CRC Handbook of Neurohypophyseal Hormone Analogs. (pp. 17-74). CRC Press, Boca Raton. #1663

  200. Lebl,M. (1987) Synthesis, purification, and stability of the neurohypophyseal hormone analogs. In K.Jost, M.Lebl & F.Brtnik (Eds.), CRC Handbook of Neurohypophyseal Hormone Analogs. (pp. 23-82). CRC Press, Boca Raton. #1658

  201. Lebl,M. (1987) Isotopically modified analogs. In K.Jost, M.Lebl & F.Brtnik (Eds.), CRC Handbook of Neurohypophyseal Hormone Analogs. (pp. 83-104). CRC Press, Boca Raton. #1659

  202. Lebl,M. & Hruby,V.J. (1987) Other methods used in the investigation of neurohypophyseal hormone analog conformations. In K.Jost, M.Lebl & F.Brtnik (Eds.), CRC Handbook of Neurohypophyseal Hormone Analogs. (pp. 155-159). CRC Press, Boca Raton. #1661

  203. Lebl,M. (1987) Modification of other functional groups. In K.Jost, M.Lebl & F.Brtnik (Eds.), CRC Handbook of Neurohypophyseal Hormone Analogs. (pp. 156-160). CRC Press, Boca Raton. #1662

  204. Lebl,M. (1987) Analogs with dissociated and/or high activities. II.Uterotonic activity. In K.Jost, M.Lebl & F.Brtnik (Eds.), CRC Handbook of Neurohypophyseal Hormone Analogs. (pp. 78-102). CRC Press, Boca Raton. #1665

  205. Lebl,M. (1987) Analogs with dissociated and/or high activities. I.Introduction. In K.Jost, M.Lebl & F.Brtnik (Eds.), CRC Handbook of Neurohypophyseal Hormone Analogs. (pp. 75-78). CRC Press, Boca Raton. #1664

  206. Lebl,M., Sugg,E.E., Van Binst,G., van der Elst,P., Tourwe,D., Slaninova,J., & Hruby,V.J. (1987) Analogs of oxytocin containing a modified peptide bond. Int. J. Peptide Prot. Res., 30, 318-322. #1767 (Available on Internet)

  207. Lebl,M., Jost,K. & Brtnik,F. (1987) Tables of analogs. In K.Jost, M.Lebl & F.Brtnik (Eds.), CRC Handbook of Neurohypophyseal Hormone Analogs. (pp. 127-268). CRC Press, Boca Raton. #1668

  208. Lebl,M., Fric,I., Sugg,E.E., Cody,W.L. & Hruby,V.J. (1987) Conformational studies of carba-analogs of oxytocin. In D.Theodoropoulos (Ed.), Peptides 1986, Proc.19.EPS. (pp. 341-344). Walter de Gruyter & Co., Berlin. #1769 (Available on Internet)

  209. Lebl,M. (1987) Analogs with dissociated and/or high activities. III. Galactogogic activity. In K.Jost, M.Lebl & F.Brtnik (Eds.), CRC Handbook of Neurohypophyseal Hormone Analogs. (pp. 102-109). CRC Press, Boca Raton. #1666

  210. Zaoral,M., Blaha,I., Lebl,M. & Barth,T. (1987) Vasopressin analogs with strong agonistic-antagonistic properties. In D.Theodoropoulos (Ed.), Peptides 1986, Proc.19.EPS. (pp. 465-468). Walter de Gruyter & Co., Berlin. #1770 (Available on Internet)

  211. Zicha,J., Kunes,J., Lebl,M., Pohlova,I., & Jelinek,J. (1987) Haemodynamics and the participation of pressor systems in young and adult rats with age-dependent doca-salt hypertension. Physiol. Bohemoslov., 36, 89-92. #1771 (Available on Internet)

  212. Hermann,P., Jannasch,R., & Lebl,M. (1986) Application of high-performance liquid chromatography and capillary isotachophoresis to the purification and characterization of products of peptide synthesis. J. Chromatogr., 351, 283-293. #1765 (Available on Internet)

  213. Hrbas,P., Barth,T., Lebl,M., Papsuevich,A.O., & Flegel,M. (1985) Mono- and diiodo-derivatives of neurohypophysial hormones and their analogues. Beitr. Wirkstofforsch., 24, 182-187. #1764 (Available on Internet)

  214. Lebl,M., Drasar,P., Koroniak,H., Milecki,J., & Ikonomov,O.C. (1985) Nejnovejsø poznatky v chemii porkanovych sloucenin. Chem. Listy, 79, 410-417. #1763 (Available on Internet)

  215. Lebl,M. (1985) Carba analogues of neurohypophysial hormones. In W.S.Hancock (Ed.), Handbook of the Use of High Performance Liquid Chromatography for the Analytical and Preparative Separation of Amino Acids, Peptides and Proteins. (pp. 169-178). CRC Press, Boca Raton. #1740 (Available on Internet)

  216. Lebl,M., Barth,T., Servitova,L., Slaninova,J., & Jost,K. (1985) Oxytocin analogues with inhibitory properties, containing in position 2 a hydrophobic amino acid of D-configuration. Collect. Czech. Chem. Commun., 50, 132-145. #1761 (Available on Internet)

  217. Lebl,M., Hruby,V.J., Slaninova,J., & Barth,T. (1985) Solid phase synthesis and biological activities of oxytocin carba analogues containing threonine in position 4. Collect. Czech. Chem. Commun., 50, 418-427. #1762 (Available on Internet)

  218. Hrbas,P., Skopkova,J., Zicha,J., Barth,T., Lebl,M., & Jost,K. (1984) Nacartocin - analogue of oxytocin with enhanced natriuretic properties: natriuretic and hemodynamic characteristics. Endocrinol. Exper., 18, 117-124. #1751 (Available on Internet)

  219. Lebl,M., Cody,W.L., & Hruby,V.J. (1984) Cyclic melanotropins. Part VI. Reverse phase HPLC studies. J. Liq. Chromatogr., 7, 1195-1210. #1752 (Available on Internet)

  220. Lebl,M., Cody,W.L., Wilkes,B.C., Hruby,V.J., Castrucci,A.M.L., & Hadley,M.E. (1984) Modification of the disulfide bridge in cyclic melanotropins. Collect. Czech. Chem. Commun., 49, 2680-2688. #1758 (Available on Internet)

  221. Lebl,M., Barth,T., Servitova,L., Slaninova,J., & Hrbas,P. (1984) Synthesis and properties of carba-6-analogues of oxytocin containing a deaminopenicillamine residue in position 1. Collect. Czech. Chem. Commun., 49, 2012-2023. #1757 (Available on Internet)

  222. Lebl,M., Cody,W.L., Wilkes,B.C., Hruby,V.J., Castrucci,A.M.L., & Hadley,M.E. (1984) Cyclic melanotropins. Part VII: Modified ring structures: Synthesis and biological activity. Int. J. Peptide Prot. Res., 24, 472-479. #1759 (Available on Internet)

  223. Lebl,M., & Hruby,V.J. (1984) Synthesis of cyclic peptides by solid phase technology. Tetrahedron Lett., 25, 2067-2068. #1708 (Available on Internet)

  224. Lebl,M., Barth,T., Crankshaw,D.J., Cerny,B., Daniel,E.E., Grover,A.K., & Jost,K. (1984) Synthesis and properties of [2-[3,5-(3)H2]-tyrosine,4-glutamic acid]deamino-1-carba-oxytocin. Collect. Czech. Chem. Commun., 49, 1921-1926. #1756 (Available on Internet)

  225. Prochazka,Z., Lebl,M., Barth,T., Hlavacek,J., Trka,A., Budesinsky,M., & Jost,K. (1984) Synthesis and properties of oxytocin analogues modified in the tripeptide side chain. Collect. Czech. Chem. Commun., 49, 642-652. #1755 (Available on Internet)

  226. Skopkova,J., Barth,T., Hrbas,P., Jost,K., & Lebl,M. (1984) Natriuretic properties of [2-p-ethylphenylalanine]deamino-6- carba-oxytocin (Nacartocin) in cats. Exp. Clin. Endocrinol., 84, 235-238. #1760 (Available on Internet)

  227. Barth,T., Cantau,B., Butlen,D., Guillon,G., Jard,S., Lebl,M., & Jost,K. (1983) Oxytocin and vasopressin analogues capable of competition with vasopressin binding to rat liver membranes. Collect. Czech. Chem. Commun., 48, 1788-1795. #1747 (Available on Internet)

  228. Barth,T., Lebl,M., Jost,K., Cantau,B., Butlan,D., Guillon,G. & Jard,S. (1983) Interactions of deamino-6-carba-oxytocin analogues in rat kidney and liver membrane systems. In K.Blaha & P.Malon (Eds.), Peptides 1982,Proc.17.EPS. (pp. 467-470). Walter de Gruyter, Berlin. #1746 (Available on Internet)

  229. Budesinsky,M., Jezek,J., Krchnak,V., Lebl,M., Zaoral,M., Rotta,J. & Straka,R. (1983) Synthetic fragments of bacterial cell walls. Physicochemical and biological properties. In K.Blaha & P.Malon (Eds.), Peptides 1982,Proc.17.EPS. (pp. 305-310). Walter de Gruyter, Berlin. #1743 (Available on Internet)

  230. Butlen,D., Barth,T., Cantau,B., Guillon,G., Jard,S., Lebl,M., Brtnik,F., & Jost,K. (1983) The structural requirements of oxytocin and vasopressin analogues for the activation of adenylate cyclase in the rat kidney medullary membrane system. Collect. Czech. Chem. Commun., 48, 3166-3176. #1748 (Available on Internet)

  231. Krojidlo,M., Flegel,M. & Lebl,M. (1983) Method for cyclization of carba analogues of oxytocin. In K.Blaha & P.Malon (Eds.), Peptides 1982,Proc.17.EPS. (pp. 199-202). Walter de Gruyter, Berlin. #1742 (Available on Internet)

  232. Lebl,M., Barth,T., Servitova,L., Slaninova,J. & Jost,K. (1983) Analogues of neurohypophysial hormones containing a D-amino acid in position 2. In K.Blaha & P.Malon (Eds.), Peptides 1982,Proc.17.EPS. (pp. 457-460). Walter de Gruyter, Berlin. #1745 (Available on Internet)

  233. Lebl,M. (1983) Analogues of neurohypophysial hormones with inhibitory effect on the pressoric activity of vasopressin. In D.F.Chebotarev & V.V.Frolkis (Eds.), Vasopressin and Pathology of the Cardiovascular System in Aging. (pp. 108-114). Institute of Gerontology, Kiev. #1750 (Available on Internet)

  234. Lebl,M. (1983) Amino acids and peptides CLXXXI. Separation of diastereoisomers of oxytocin analogues. J. Chromatogr., 264, 459-462. #1749 (Available on Internet)

  235. Lebl,M., & Gut,V. (1983) Calculation of the rate constant of a reversible reaction from the chromatographic peaks for muranyl dipeptide anomers. J. Chromatogr., 260, 478-482. #1741 (Available on Internet)

  236. Lebl,M. & Barth,T. (1983) Synthesis and some activities of [1-penicillamine]deamino-6-carba-oxytocin. In V.J.Hruby & D.H.Rich (Eds.), Peptides:Structure and Function,Proc.8.APS. (pp. 357-360). Pierce, Rockford. #1753 (Available on Internet)

  237. Prochazka,Z., Lebl,M., Barth,T., Hlavacek,J. & Jost,K. (1983) Two analogues of oxytocin with modified proline cyclic structure. In K.Blaha & P.Malon (Eds.), Peptides 1982,Proc.17.EPS. (pp. 441-444). Walter de Gruyter, Berlin. #1744 (Available on Internet)

  238. Lebl,M., Pospisek,J., Hlavacek,J., Barth,T., Malon,P., Servitova,L., Hauzer,K., & Jost,K. (1982) Analogues of neurohypophysial hormones containing tert.leucine: synthesis and properties. Collect. Czech. Chem. Commun., 47, 689-701. #1737 (Available on Internet)

  239. Lebl,M., Hrbas,P., Skopkova,J., Slaninova,J., Machova,A., Barth,T., & Jost,K. (1982) Synthesis and properties of oxytocin analogues with high and selective natriuretic activity. Collect. Czech. Chem. Commun., 47, 2540-2560. #1739 (Available on Internet)

  240. Lebl,M. (1982) Correlation between hydrophobicity of substituents in the phenylalanine moiety of oxytocin carba-analogues and reversed- phase-chromatographic k' values. J. Chromatogr., 242, 342-345. #1738 (Available on Internet)

  241. Barth,T., Hrbas,P., Skopkova,J., Slaninova,J., Lebl,M. & Jost,K. (1981) Natriuretic effects of oxytocin analogues. In K.Brunfeldt (Ed.), Peptides 1980,Proc.16.EPS. (pp. 416-419). Scriptor, Copenhagen. #1732 (Available on Internet)

  242. Barth,T., Slaninova,J., Servitova,L., Lebl,M., Kotsira-Engonopoulos,C., Tzougraki,C., Photaki,I., Krojidlo,M., & Jost,K. (1981) The effect of some structural modification of the oxytocin molecule on the duration of the galactogogic response. Collect. Czech. Chem. Commun., 46, 2441-2445. #1736 (Available on Internet)

  243. Bienert,M., Lebl,M., Mehlis,B. & Niedrich,H. (1981) Synthesis and application of methionin S-tert-butylsulfonium peptides. In K.Brunfeldt (Ed.), Peptides 1980,Proc.16.EPS. (pp. 127-132). Scriptor, Copenhagen. #1731 (Available on Internet)

  244. Lebl,M., Barth,T. & Jost,K. (1981) Chromatographic and pharmacological properties of carba- analogues of neurohypophyseal hormones sulfoxides. A general method of sulfoxide group determination in peptides. In K.Brunfeldt (Ed.), Peptides 1980,Proc.16.EPS. (pp. 719-724). Scriptor, Copenhagen. #1733 (Available on Internet)

  245. Prochazka,Z., Lebl,M., Servitova,L., Barth,T., & Jost,K. (1981) Synthesis and pharmacological properties of 2-p-fluorophenyl- alanine deamino-1-carba-oxytocin and of its diastereoisomeric sulfoxides. Collect. Czech. Chem. Commun., 46, 947-956. #1734 (Available on Internet)

  246. Slaninova,J., Lebl,M., Barth,T., & Jost,K. (1981) The effect of magnesium ions on the uterotonic activity of carba analogues of oxytocin modified in position 4. Collect. Czech. Chem. Commun., 46, 1689-1692. #1735 (Available on Internet)

  247. Barth,T., Slaninova,J., Lebl,M., & Jost,K. (1980) Biological activities and protracted action of carba-analogues of deamino-oxytocin with O-methyltyrosine in position 2. Collect. Czech. Chem. Commun., 45, 3045-3050. #1728 (Available on Internet)

  248. Hrbas,P., Barth,T., Skopkova,J., Lebl,M., & Jost,K. (1980) Effect of some oxytocin analogues on natriuresis in rats. Endocrinol. Exper., 14, 151-157. #1723 (Available on Internet)

  249. Hrbas,P., Skopkova,J., Barth,T., Lebl,M. & Jost,K. (1980) Renal sodium excretion in rats. Effect of amino acid replacement in position 4 of the oxytocin molecule. In B.Lichardus, R.W.Schrier & J.Ponec (Eds.), Hormonal Regulation of Sodium Excretion. (pp. 169-172). Elsevier, Amsterdam. #1730 (Available on Internet)

  250. Lebl,M., Machova,A., Hrbas,P., Barth,T., & Jost,K. (1980) Analogues of deamino-1-carba-oxytocin with aliphatic amino acid in position 4: Chemical synthesis and biological activities. Collect. Czech. Chem. Commun., 45, 2714-2723. #1724 (Available on Internet)

  251. Lebl,M., Barth,T., Skopkova,J., & Jost,K. (1980) Synthesis and some pharmacological properties of [7-glycine,8- ornithine]-vasopressin and of its two analogues. Collect. Czech. Chem. Commun., 45, 2865-2871. #1726 (Available on Internet)

  252. Lebl,M. (1980) High-performance liquid chromatography of carba analogues of oxytocin; a method for the determination of sulfides and sulfoxides in peptides. Collect. Czech. Chem. Commun., 45, 2927-2937. #1727 (Available on Internet)

  253. Lebl,M., Barth,T., & Jost,K. (1980) Synthesis and pharmacological properties of oxytocin analogues modified simultaneously in position 2 and in the disulfide bridge. Collect. Czech. Chem. Commun., 45, 2855-2864. #1725 (Available on Internet)

  254. Skopkova,J., Hrbas,P., Barth,T., Lebl,M. & Jost,K. (1980) Renal sodium excretion in rats. Effect of structural modification of position 2 of deamino-6-carba-oxytocin. In B.Lichardus, R.W.Schrier & J.Ponec (Eds.), Hormonal Regulation of Sodium Secretion. (pp. 163-168). Elsevier, Amsterdam. #1729 (Available on Internet)

  255. Barth,T., Lebl,M., Bojanovska,V. & Jost,K. (1979) Analogues of oxytocin acting as irreversible inhibitors of oxytocin. In I.Z.Siemion & G.Kupryszewski (Eds.), Peptides 1978,Proc.15.EPS. (pp. 475-479). Wroclaw University Press, Wroclaw. #1722 (Available on Internet)

  256. Lebl,M. & Jost,K. (1979) Selective oxidation of sulfur in peptide synthesis. In I.Z.Siemion & G.Kupryszewski (Eds.), Peptides 1978,Proc.15.EPS. (pp. 109-112). Wroclaw University Press, Wroclaw. #1721 (Available on Internet)

  257. Lebl,M., Barth,T., & Jost,K. (1979) Analogues of oxytocin with esters of glutamic acid instead of glutamine in position 4: synthesis of a compound with high and specific galactogogic activity. Collect. Czech. Chem. Commun., 44, 2563-2572. #1719 (Available on Internet)

  258. Lebl,M., Bojanovska,V., Barth,T., & Jost,K. (1979) Synthesis and properties of oxytocin analogues acting as irreversible inhibitors of the uterotonic response to oxytocin. Collect. Czech. Chem. Commun., 44, 2573-2582. #1720 (Available on Internet)

  259. Lebl,M., Dimeli,A., Bojanovska,V., Slaninova,J., Barth,T., & Jost,K. (1979) Synthesis and some biological properties of amides derived from [4-glutamic acid]deamino-1-carba-oxytocin. Collect. Czech. Chem. Commun., 44, 2556-2562. #1718 (Available on Internet)

  260. Lebl,M., Barth,T., & Jost,K. (1978) Na-glycyl-glycyl-glycyl-8-ornithine-vasopressin: A trypsin resistant vasopressin analog with a specific pressor effect. Collect. Czech. Chem. Commun., 43, 1300-1305. #1715 (Available on Internet)

  261. Lebl,M., Barth,T., & Jost,K. (1978) Synthesis, reduction, and pharmacological properties of the sulfoxides of some carba-analogues of oxytocin. Collect. Czech. Chem. Commun., 43, 1538-1556. #1716 (Available on Internet)

  262. Lebl,M., & Jost,K. (1978) Mechanismus racemisace derivßtu aminokyselin. Chem. Listy, 72, 252-266. #1713 (Available on Internet)

  263. Lebl,M., Bojanovska,V., Barth,T., & Jost,K. (1978) Oxytocin analogs effective as noncompetitive inhibitors in uterotonic test. Experientia, 34, 1543-1544. #1717 (Available on Internet)

  264. Lebl,M., & Jost,K. (1978) Synthesis of [4-glutamic acid]deamino-1-carba-oxytocin. Collect. Czech. Chem. Commun., 43, 523-534. #1714 (Available on Internet)

  265. Ferles,M., Kocian,O., Lebl,M., Lovy,J., Radl,S., Silhankova,A., & Stern,P. (1976) Electrolytic reduction of quarternary salts of some alcohols of pyridine series, of corresponding alkylpyridines and alkenylpyridines. Collect. Czech. Chem. Commun., 41, 598-603. #1712 (Available on Internet)

  266. Ferles,M., Lebl,M., Stern,P., & Trska,P. (1975) Mixed electrolytic reduction of 1,4,-dimethylpyridinium methylsulfate with acetone and of 1-methylpyridinium methylsulfate with cyclopentanone. Collect. Czech. Chem. Commun., 40, 2183-2190. #1711 (Available on Internet)

  267. Ferles,M., Lebl,M., Silhankova,A., Stern,P., & Wimmer,Z. (1975) Reduction of tertiary alcohols of the pyridine series and corresponding alkenylpyridines with zinc and formic acid. Collect. Czech. Chem. Commun., 40, 1571-1575. #1710 (Available on Internet)