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PAPERS PUBLISHED IN 1997

This list is arranged by the name of the first author. Please, note the change in numbering of the references. Any omissions, mistakes and inconsistencies please communicate to the authors of compilation (michal@5z.com). (If you are pointing to any reference, please use its ID# -- the last number in the reference.) You are welcome to use this compilation in your work. Proper way to quote it in your paper is: Lebl M., Leblova Z.: Dynamic database of references in molecular diversity. Internet http://www.5z.com.


Recently added entries are marked in bold

  1. Anonymous. (1997) Combinatorial chemistry. Chemtech, 27, 3-3. #9395

  2. Anonymous. (1997) Combinatorial chemistry to develop new drugs. Canc. J. Sci. Amer., 3, 312-313. #9888

  3. Abraham, D. (1997) Combining legal and business strategies to develop combinatorial chemistry businesses. Nat. Biotech., 15, 679-682. #9358

  4. Adamczyk, M., Gebler, J.C., & Grote, J. (1997) The utility of enzymes in generating molecular diversity. Lipase mediated amidation of polybenzyl esters. Bioorg. Med. Chem. Lett., 7, 1027-1030. #10085

  5. Adams, E., Basten, A., Rodda, S., & Britton, W.J. (1997) Human T-cell clones to the 70-kilodalton heat shock protein of mycobacterium leprae define myobacterium-specific epitopes rather than shaped epitopes. Infec. Immunity, 65, 1061-1070. #9550

  6. Adey, N.B., & Kay, B.K. (1997) Isolation of peptides from phage-displayed random peptide libraries that interact with the talin-binding domain of vinculin. Biochem. J., 324, 523-528. #9190

  7. Agrafiotis, D.K. (1997) Stochastic algorithms for maximizing molecular diversity. Journal of Chemical Information and Computer Sciences, 37, 841-851. #8721

  8. Akada, R., Yamamoto, J., & Yamashita, I. (1997) Screening and identification of yeast sequences that cause growth inhibition when overexpressed. Mol. Gen. Genet., 254, 267-274. #12481

  9. Akaji, K., & Kiso, Y. (1997) Macrocyclization on solid support using Heck reaction. Tetrahedron Lett., 38, 5185-5188. #9035

  10. Alajoki, M.L., Baxter, G.T., Bemiss, W.R., Blau, D., Bousse, L.J., Chan, S.D.H., Dawes, T.D., Hahnenberger, K.M., Hamilton, J.M., Lam, P., McReynolds, R.J., Modlin, D.N., Owicki, J.C., Parce, J.W., Redington, D., Stevenson, K., Wada, H.G. & Williams, J. (1997) High-performance microphysiometry in drug discovery. In J.P. Devlin (Ed.), High Throughput Screening: The Discovery of Bioactive Substances. (pp. 427-442). Marcel Dekker,Inc., New York. #9011

  11. Allee, C. (1997) Systems integration. In J.P. Devlin (Ed.), High Throughput Screening: The Discovery of Bioactive Substances. (pp. 583-598). Marcel Dekker,Inc., New York. #9022

  12. Ammosova, T.N., Ouporov, I.V., Rubtsova, M.Y., Ignatenko, O.V., Egorov, A.M., Kolesanova, E.F., & Archakov, A.I. (1997) Epitope mapping of horseradish peroxidase (isoenzyme C). Biochemistry-Engl. Tr., 62, 440-447. #9217

  13. An, H.Y., Cummins, L.L., Griffey, R.H., Bharadwaj, R., Haly, B.D., Fraser, A.S., Wilson-Lingardo, L., Risen, L.M., Wyatt, J.R., & Cook, P.D. (1997) Solution phase combinatorial chemistry: Discovery of novel polyazapyridinophanes with potent antibacterial activity by a solution phase simultaneous addition of functionalities approach [review]. J. Amer. Chem. Soc., 119, 3696-3708. #9137

  14. An, H.Y., Haly, B.D., Fraser, A.S., Guinosso, C.J., & Cook, P.D. (1997) Solution phase combinatorial chemistry. Synthesis of novel linear pyridinopolyamine libraries with potent antibacterial activity. J. Org. Chem., 62, 5156-5164. #9440

  15. Anand, N., Jain, S., & Sinha, N. (1997) Molecular diversity generation through reactive lactams. J. Ind. Chem. Soc., 74, 948-954. #10989

  16. Armstrong, R.W., Brown, S.D., Keating, T.A. & Tempest, P.A. (1997) Combinatorial synthesis exploiting multiple-component condensations, microchip encoding, and resin capture. In S.R. Wilson & A.W. Czarnik (Eds.), Combinatorial Chemistry. Synthesis and Application. (pp. 153-190). John Wiley & Sons,Inc., New York. #8357

  17. Arnau, J., & Sorensen, K.I. (1997) The isolation of novel heat shock genes in Lactococcus lactis using RNA subtractive hybridization. Gene, 188, 229-234. #12482

  18. Arnold, D., Keilholz, W., Schild, H., Dumrese, T., Stevanovic, S., & Rammensee, H.G. (1997) Substrate specificity of cathepsins D and E determined by N-terminal and C-terminal sequencing of peptide pools. Eur. J. Biochem., 249, 171-179. #10103

  19. Arumugam, V., Routledge, A., Abell, C., & Balasubramanian, S. (1997) Synthesis of 2-oxindole derivatives via the intramolecular Heck reaction on solid support. Tetrahedron Lett., 38, 6473-6476. #9321

  20. Arya, P., & Ben, R.N. (1997) Combinatorial chemistry for the synthesis of carbohydrate libraries. Angew. Chem. Int. Ed., 36, 1280-1282. #9481

  21. Arza, B., Felez, J., Lopezalemany, R., Miles, L.A., & Munozcanoves, P. (1997) Identification of an epitope of alpha-enolase (a candidate plasminogen receptor) by phage display. Thromb. Haemost., 78, 1097-1103. #10106

  22. Atrash, B., & Bradley, M. (1997) A pH cleavable linker for zone diffusion assays and single bead solution screens in combinatorial chemistry. Chem. Commun., 1397-1398. #9527

  23. Aujame, L., Sodoyer, R., & Teillaud, J.L. (1997) Phage display and antibody engineering: A French overview. Trends Biotech., 15, 155-157. #10462

  24. Avalle, B., Vanwetswinkel, S., & Fastrez, J. (1997) In vitro selection for catalytic turnover from a library of beta-lactamase mutants and penicilin-binding proteins. Bioorg. Med. Chem. Lett., 7, 479-484. #10022

  25. Babiak, J. (1997) Management and service issues of a centralized robotic HTS core. In J.P. Devlin (Ed.), High Throughput Screening: The Discovery of Bioactive Substances. (pp. 461-470). Marcel Dekker,Inc., New York. #9014

  26. Babiak, J. Transforming your robotics into an infrastructure for the future. In: Anonymous. (Eds.) Zymark Corporation, Hopkington, MA p.35 Proceedings of the International Symposium on Laboratory Automation and Robotics 1996. #8282

  27. Baca, M., Scanlan, T.S., Stephenson, R.C., & Wells, J.A. (1997) Phage display of a catalytic antibody to optimize affinity for transition-state analog binding. Proc. Natl. Acad. Sci. USA, 94, 10063-10068. #10107

  28. Backes, B.J., & Ellman, J.A. (1997) Solid support linker strategies. Curr. Opin. Chem. Biol., 1, 86-93. #8746

  29. Bailey, N., Cooper, A.W.J., Deal, M.J., Dean, A.W., Gore, A.L., Hawes, M.C., Judd, D.B., Merritt, A.T., Storer, R., Travers, S., & Watson, S.P. (1997) Solution-phase combinatorial chemistry in lead discovery. Chimia, 51, 832-837. #9733

  30. Balass, M., Katchalski-Katzir, E., & Fuchs, S. (1997) The alpha-bungarotoxin binding site on the nicotinic acetylcholine receptor: Analysis using a phage-epitope library. Proc. Natl. Acad. Sci. USA, 94, 6054-6058. #9188

  31. Balcer-Kubiczek, E.K., Meltzer, S.J., Han, L.H., Zhang, X.F., Shi, Z.M., Harrison, G.H., & Abraham, J.M. (1997) Csa-19, a radiation-responsive human gene, identified by an unbiased two-gel cDNA library screening method in human cancer cells. Oncogene, 14, 3051-3057. #12483

  32. Balding, D.J., & Torney, D.C. (1997) The design of pooling experiments for screening a clone map. Fungal Genet. Biol., 21, 302-307. #12484

  33. Baldino, C.M., Casebier, D.S., Caserta, J., Slobodkin, G., Tu, C., & Coffen, D.L. (1997) Convergent parallel synthesis. Synlett, 488-490. #9077

  34. Baldwin, J.J. & Dolle, R. (1997) Deconvolution tools for solid-phase synthesis. In A.W. Czarnik & S.H. DeWitt (Eds.), A Practical Guide to Combinatorial Chemistry. (pp. 153-174). American Chemical Society, Washington,DC. #11698

  35. Baldwin, J.J. & Henderson, I. (1997) Synthesis of encoded small molecule combinatorial libraries via ECLiPS. In J.P. Devlin (Ed.), High Throughput Screening: The Discovery of Bioactive Substances. (pp. 167-190). Marcel Dekker,Inc., New York. #8993

  36. Baldwin, J.J. & Dolle, R.E. (1997) Deconvolution methods in solid-phase synthesis. In W.H. Moos, M.R. Pavia, B.K. Kay & A.D. Ellington (Eds.), Annual Reports in Combinatorial Chemistry and Molecular Diversity. (pp. 287-297). ESCOM, Leiden. #8629

  37. Banks, M., Fogarty, S., Valler, M., Mills, K., O'Brien, S., Binnie, A., and Houston, J. Automated high throughput screening to aid the drug hunter at Glaxo Wellcome. In: Anonymous. (Eds.) Zymark Corporation, Hopkington, MA p.220 Proceedings of the International Symposium on Laboratory Automation and Robotics 1996. #8306

  38. Banville, S. C. and Zuckermann, R. N. Accelerating drug discovery by high-throughput combinatorial synthesis. In: Anonymous. (Eds.) Zymark Corporation, Hopkington, MA p.77 Proceedings of the International Symposium on Laboratory Automation and Robotics 1996. #8285

  39. Barany, G., Albericio, F., Kates, S.A., & Kempe, M. (1997) Polyethylene glycol-containing supports for solid phase synthesis of peptides and combinatorial organic libraries. Polym. Preprint., 38, 587-588. #8520

  40. Barany, G., Albericio, F., Kates, S.A., & Kempe, M. (1997) Poly(ethylene glycol)-containing supports for solid-phase synthesis of peptides and combinatorial organic libraries. ACS Symp. Ser., 680, 239-264. #9612

  41. Barany, G. & Kempe, M. (1997) The contex of solid-phase synthesis. In A.W. Czarnik & S.H. DeWitt (Eds.), A Practical Guide to Combinatorial Chemistry. (pp. 51-97). American Chemical Society, Washington,DC. #11696

  42. Barnard, J.M., & Downs, G.M. (1997) Computer representation and manipulation of combinatorial libraries [review]. Perspect. Drug Disc. Design, 7-8, 13-30. #10724

  43. Bastien, N., Trudel, M., & Simard, C. (1997) Protective immune responses induced by the immunization of mice with a recombinant bacteriophage displaying an epitope of the human respiratory syncytial virus. Virology, 234, 118-122. #9444

  44. Bauer, B.E. (1997) Database systems. In J.P. Devlin (Ed.), High Throughput Screening: The Discovery of Bioactive Substances. (pp. 551-582). Marcel Dekker,Inc., New York. #9021

  45. Bauer, U., Ho, W.B., & Koskinen, A.M.P. (1997) A novel linkage for the solid-phase synthesis of hydroxamic acids. Tetrahedron Lett., 38, 7233-7236. #9563

  46. Baxter, A.D. (1997) Meeting client needs in combinatorial chemistry: A service company perspective. Drug Disc. Today, 2, 307-308. #9429

  47. Baxter, A.D. (1997) Synthesis utilizing insoluble polymers: New reactions and small molecules. Curr. Opin. Chem. Biol., 1, 79-85. #8739

  48. Beggs, M. Use of a two armed Zymark robot for high throughput screening. In: Anonymous. (Eds.) Zymark Corporation, Hopkington, MA p.206 Proceedings of the International Symposium on Laboratory Automation and Robotics 1996. #8305

  49. Beggs, M. & Major, J.S. (1997) Flexible use of people and machines. In J.P. Devlin (Ed.), High Throughput Screening: The Discovery of Bioactive Substances. (pp. 471-482). Marcel Dekker,Inc., New York. #9015

  50. Beggs, M. (1997) Use of a two-armed Zymark robot for high throughput screening. J. Biomol. Screen., 2, 71-78. #9841

  51. Bellott, E.M., Bondaryk, R., & Luther, A.L. (1997) Combinatorial chemistry in the drug discovery process. Clin. Res. Regul. Affairs, 14, 231-241. #12202

  52. Benecke, C., Gruner, T., Kerber, A., Laue, R., & Wieland, T. (1997) Molecular structure generation with molgen, new features and future developments. Fresenius J. Anal. Chem., 359, 23-32. #10116

  53. Benkovic, S., Miller, G.P., Zong, W. & Smiley, J. (1997) Combinatorial libraries of peptides, proteins, and antibodies using biological systems. In S.R. Wilson & A.W. Czarnik (Eds.), Combinatorial Chemistry. Synthesis and Application. (pp. 241-260). John Wiley & Sons,Inc., New York. #8361

  54. Beresini, M.H., Sadick, M.D., Galloway, A.L., Yen, R., Yeh, S.H., Chang, A.C., Shelton, D.L. & Wong, W.L.T. (1997) Assays for small molecule agonists and antagonists of the neurotrophin receptors. In J.P. Devlin (Ed.), High Throughput Screening: The Discovery of Bioactive Substances. (pp. 329-344). Marcel Dekker,Inc., New York. #9004

  55. Berk, S.C., & Chapman, K.T. (1997) Spatially arrayed mixture (SPAM) technology: Synthesis of two-dimensionally indexed orthogonal combinatorial libraries. Bioorg. Med. Chem. Lett., 7, 837-842. #9256

  56. Berlin, K., Jain, R.K., Tetzlaff, C., Steinbeck, C., & Richert, C. (1997) Spectrometrically monitored selection experiments: Quantitative laser desorption mass spectrometry of small chemical libraries. Chem. Biol., 4, 63-77. #8400

  57. Beutel, B.A. (1997) Discovery and identification of lead compounds from combinatorial mixtures. Annu. Rep. Med. Chem., 32, 261-268. #9698

  58. Bhagwat, S.S., & Williams, M. (1997) P2 purine and pyrimidine receptors: Emerging superfamilies of G-protein-coupled and ligand-gated ion channel receptors [review]. Eur. J. Med. Chem., 32, 183-193. #9244

  59. Bhalay, G., Blaney, P., Palmer, V.H., & Baxter, A.D. (1997) Solid-phase synthesis of diverse tetrahydro-1,4-benzodiazepine-2-ones. Tetrahedron Lett., 38, 8375-8378. #9674

  60. Biebricher, C.K., & Gardiner, W.C. (1997) Molecular evolution of RNA in vitro. Biophys. Chem., 66, 179-192. #10119

  61. Birkenmeier, G., Osman, A.A., Kopperschlager, G., & Mothes, T. (1997) Epitope mapping by screening of phage display libraries of a monoclonal antibody directed against the receptor binding domain of human alpha-2-macroglobulin. FEBS Lett., 416, 193-196. #10120

  62. Bishop, A.C., Moore, D., Scanlan, T.S., & Shokat, K.M. (1997) Screening a hydroxystilbene library for selective inhibition of the b cell antigen receptor kinase cascade. Tetrahedron, 53, 11995-12004. #10121

  63. Bitan, G., Sukhotinsky, I., Mashriki, Y., Hanani, M., Selinger, Z., & Gilon, C. (1997) Synthesis and biological activity of novel backbone-bicyclic substance-P analogs containing lactam and disulfide bridges. J. Pept. Res., 49, 421-426. #9198

  64. Blackburn, C., Pingali, A., Kehoe, T., Herman, L.W., Wang, H.Q., & Kates, S.A. (1997) Libraries of angiotensin converting enzyme inhibitors: Solid-phase synthesis and affinity selection. Bioorg. Med. Chem. Lett., 7, 823-826. #9255

  65. Blackburn, C., & Kates, S.A. (1997) Solid-phase synthesis of cyclic homodetic peptides. Methods Enzymol., 289, 175-198. #9857

  66. Blackburn, C., Albericio, F., & Kates, S.A. (1997) Functionalized resins and linkers for solid-phase synthesis of small molecules. Drugs Future, 22, 1007-1025. #9840

  67. Blanchard, B.J., Konopka, G., Russell, M., & Ingram, V.M. (1997) Mechanism and prevention of neurotoxicity caused by beta-amyloid peptides: Relation to Alzheimer's-disease. Brain Res., 776, 40-50. #10122

  68. Blaney, J.M., & Martin, E.J. (1997) Computational approaches for combinatorial library design and molecular diversity analysis. Curr. Opin. Chem. Biol., 1, 54-59. #8715

  69. Bloxham, D. P. The current status and future of drug discovery. In: W. Hori. (Eds.) 1996; International Business Communications,Inc., Southborough p.7.4.1 #8890

  70. Boder, E.T., & Wittrup, K.D. (1997) Yeast surface display for screening combinatorial polypeptide libraries. Nat. Biotech., 15, 553-557. #9194

  71. Boger, D.L., Chai, W., Ozer, R.S., & Andersson, C.M. (1997) Solution-phase combinatorial synthesis via the olefin metathesis reaction. Bioorg. Med. Chem. Lett., 7, 463-468. #10021

  72. Boger, D.L., Ozer, R.S., & Andersson, C.M. (1997) Generation of targeted C(2)-symmetrical compound libraries by solution-phase combinatorial chemistry. Bioorg. Med. Chem. Lett., 7, 1903-1908. #9425

  73. Bojanic, D., Keighley, W.W., Russell, M.J. & Wood, T.P. (1997) Factors for the successful integration of assays, equipment, robotics, and software. In J.P. Devlin (Ed.), High Throughput Screening: The Discovery of Bioactive Substances. (pp. 493-508). Marcel Dekker,Inc., New York. #9017

  74. Bolton, G.L., Hodges, J.C., & Rubin, J.R. (1997) Solid phase synthesis of fused bicyclic amino acid derivatives via intramolecular Pauson-Khand cyclization: Versatile scaffolds for combinatorial chemistry. Tetrahedron, 53, 6611-6634. #8636

  75. Bone, R. & Salemme, F.R. (1997) The integration of structure-based design and directed combinatorial chemistry for new pharmaceutical discovery. In P. Veerapandian (Ed.), Structure-Based Drug Design. (pp. 525-539). Marcel Dekker, New York. #11242

  76. Bonnycastle, L.L., Brown, K.L., Tang, J., & Scott, J.K. (1997) Assaying phage-borne peptides by phage capture on fibrinogen or streptavidin. Biol. Chem., 378, 509-515. #10475

  77. Boojamra, C.G., Burow, K.M., Thompson, L.A., & Ellman, J.A. (1997) Solid-phase synthesis of 1,4-benzodiazepine-2,5-diones. Library preparation and demonstration of synthesis generality. J. Org. Chem., 62, 1240-1256. #8522

  78. Booth, R.J., & Hodges, J.C. (1997) Polymer-supported quenching reagent for parallel purification. J. Amer. Chem. Soc., 119, 4882-4886. #8643

  79. Borchardt, A., Liberles, S.D., Biggar, S.R., Crabtree, G.R., & Schreiber, S.L. (1997) Small molecule-dependent genetic selection in stochastic nanodroplets as a means of detecting protein-ligand interactions on a large scale. Chem. Biol., 4, 961-968. #10124

  80. Bottger, A., Bottger, V., Garcia-Echeverria, C., Chene, P., Hochkeppel, H.K., Sampson, W., Ang, K., Howard, S.F., Picksley, S.M., & Lane, D.P. (1997) Molecular characterization of the hdm2-p53 interaction. J. Mol. Biol., 269, 744-756. #10470

  81. Boumrah, D., Campbell, M.M., Fenner, S., & Kinsman, R.G. (1997) Spacer molecules in peptide sequences: Incorporation into analogues of atrial natriuretic factor. Tetrahedron, 53, 6977-6992. #9106

  82. Boutin, J.A., Gesson, I., Henlin, J.M., Bertin, S., Lambert, P.H., Volland, J.P., & Fauchere, J.L. (1997) Limitations of the coupling of amino acid mixtures for the preparation of equimolar peptide libraries. Mol. Diversity, 3, 43-60. #10098

  83. Bozicevic, K. (1997) Patent strategies in molecular diversity. In W.H. Moos, M.R. Pavia, B.K. Kay & A.D. Ellington (Eds.), Annual Reports in Combinatorial Chemistry and Molecular Diversity. (pp. 298-313). ESCOM, Leiden. #8630

  84. Bradley, E.K., Kerr, J.M., Richter, L.S., Figliozzi, G.M., Goff, D.A., Zuckermann, R.N., Spellmeyer, D.C., & Blaney, J.M. (1997) NMR structural characterization of oligo-N-substituted glycine lead compounds from a combinatorial library. Mol. Diversity, 3, 1-15. #10096

  85. Brady, P.A., & Sanders, J.K. (1997) Selection approaches to catalytic systems [review]. Chem. Soc. Rev., 26, 327-336. #10126

  86. Brandt, D.W. (1997) Multiplexed nanoliter transfers for high throughput drug screening using the Biomek 2000 and the high density replicating tool. J. Biomol. Screen., 2, 111-116. #9843

  87. Bray, A.M. (1997) Multiple peptide synthesis with commercially available Multipin kits. In I. Lefkovits (Ed.), Immunology Methods Manual. (pp. 809-816). Academic Press, San Diego. #9738

  88. Breaker, R.R. (1997) In vitro selection of catalytic polynucleotides. Chem. Rev., 97, 371-390. #8565

  89. Breaker, R.R. (1997) DNA aptamers and DNA enzymes. Curr. Opin. Chem. Biol., 1, 26-31. #8712

  90. Bristol, J.A. (1997) Applications of solid-supported organic synthesis in combinatorial chemistry: Preface. Tetrahedron, 53, xiii-xiii. #9112

  91. Broughton, H.B. (1997) Molecular modeling. Curr. Opin. Chem. Biol., 1, 392-398. #10127

  92. Brown, A.R., Rees, D.C., Rankovic, Z., & Morphy, J.R. (1997) Synthesis of tertiary amines using a polystyrene (REM) resin. J. Amer. Chem. Soc., 119, 3288-3295. #9152

  93. Brown, B.A., Cain, M., Broadbent, J., Tompkins, S., Henrich, G., Joseph, R., Casto, S., Harney, H., Greene, R., Delmondo, R. & Ng, S. (1997) FlashPlate(TM) technology. In J.P. Devlin (Ed.), High Throughput Screening: The Discovery of Bioactive Substances. (pp. 317-328). Marcel Dekker,Inc., New York. #9003

  94. Brown, D. (1997) Future pathways for combinatorial chemistry. Mol. Diversity, 2, 217-222. #8869

  95. Brown, E.G., & Nuss, J.M. (1997) Alkylation of Rink's amide linker on polystyrene resin: A reductive amination approach to modified amine-linkers for the solid phase synthesis of N-substituted amide derivatives. Tetrahedron Lett., 38, 8457-8460. #9691

  96. Brown, P.J., Smitholiver, T.A., Charifson, P.S., Tomkinson, N.C., Fivush, A.M., Sternbach, D.D., Wade, L.E., Orband-Miller, L.A., Parks, D.J., Blanchard, S.G., Kliewer, S.A., Lehmann, J.M., & Willson, T.M. (1997) Identification of peroxisome proliferator-activated receptor ligands from a biased chemical library. Chem. Biol., 4, 909-918. #10129

  97. Brown, P.J., Hurley, K.P., Stuart, L.W., & Willson, T.M. (1997) Generation of secondary alkyl amines on solid support by borane reduction: Application to the parallel synthesis of PPAR ligands. Synthesis-Stuttgart, 778-782. #9411

  98. Brown, R.D., & Martin, Y.C. (1997) The information content of 2D and 3D structural descriptors relevant to ligand-receptor binding. Journal of Chemical Information and Computer Sciences, 37, 1-9. #8717

  99. Brown, R.D., & Martin, Y.C. (1997) Designing combinatorial library mixtures using a genetic algorithm. J. Med. Chem., 40, 2304-2313. #9457

  100. Brown, R.D. (1997) Descriptors for diversity analysis [review]. Perspect. Drug Disc. Design, 7-8, 31-49. #10725

  101. Brown, R.K. & Proulx, A. (1997) Accelerating the discovery process with automation and robotics: A sure bet or a risky venture? In J.P. Devlin (Ed.), High Throughput Screening: The Discovery of Bioactive Substances. (pp. 509-524). Marcel Dekker,Inc., New York. #9018

  102. Brown, S.D., & Armstrong, R.W. (1997) Parallel synthesis of tamoxifen and derivatives on solid support via resin capture. J. Org. Chem., 62, 7076-7077. #9630

  103. Bruice, T.W., & Lima, W.F. (1997) Control of complexity constraints on combinatorial screening for preferred oligonucleotide hybridization sites on structured RNA. Biochemistry, 36, 5004-5019. #9252

  104. Bruno, J.G., Chang, M.N., Choisledeski, Y.M., Green, D.M., Mcgarry, D.G., Regan, J.R., & Volz, F.A. (1997) Synthesis of functionalized aromatic oligomers from a versatile diphenylmethane template. J. Org. Chem., 62, 5174-5190. #9441

  105. Bunin, B.A., Plunkett, M.J., Ellman, J.A., & Bray, A.M. (1997) The synthesis of a 1680 member 1,4-benzodiazepine library. New J. Chem., 21, 125-130. #9068

  106. Burbaum, J.J., & Sigal, N.H. (1997) New technologies for high-throughput screening. Curr. Opin. Chem. Biol., 1, 72-78. #8738

  107. Burger, M.T., & Still, W.C. (1997) Simple structural requirements for sequence-selective peptide receptors: Tripeptide binding by a podand ionophore. J. Org. Chem., 62, 4785-4790. #9469

  108. Burgess, K., Li, W., Linthicum, D.S., Ni, Q., Pledger, D., Rothman, R.B., & Shitangkoon, A. (1997) Libraries of opiate and anti-opiate peptidomimetics containing 2,3-methanoleucine. Bioorg. Med. Chem., 5, 1867-1871. #10131

  109. Burgess, K., Ibarzo, J., Linthicum, D.S., Russell, D.H., Shin, H., Shitangkoon, A., Totani, R., & Zhang, A.J. (1997) Solid phase syntheses of oligoureas. J. Amer. Chem. Soc., 119, 1556-1564. #8395

  110. Burgess, K., Lim, D., Bois-Choussy, M., & Zhu, J. (1997) Rapid and efficient solid phase syntheses of cyclic peptides with endocyclic biaryl ether bonds. Tetrahedron Lett., 38, 3345-3348. #8804

  111. Burioni, R., Plaisant, P., Dellicarri, V., Vannini, A., Spanu, T., Clementi, M., Fadda, G., & Varaldo, P.E. (1997) An improved phage display vector for antibody repertoire cloning by construction of combinatorial libraries. Res. Virol., 148, 161-164. #9277

  112. Burmeister, J., Von Kiedrowski, G., & Ellington, A.D. (1997) Cofactor-assisted self-cleavage in DNA libraries with a 3'-5'-phosphoramidate bond. Angew. Chem. Int. Ed., 36, 1321-1324. #12485

  113. Byk, G., Frederic, M., & Scherman, D. (1997) One pot synthesis of unsymetrically functionalized polyamines by a solid phase startegy starting from their symmetrical polyamine-counterparts. Tetrahedron Lett., 38, 3219-3222. #8798

  114. Byrgesen, E., Nielsen, J., Willert, M., & Bols, M. (1997) Combinatorial chemistry of piperidine based carbohydrate mimics. Tetrahedron Lett., 38, 5697-5700. #9412

  115. C&EN. (1997) Unique excitation emission forms basis of new taggants. C&EN, 75, 24. #8728

  116. Cabilly, S. (1997) Combinatorial Peptide Library Protocols. Humana Press, Inc., Totowa. ISBN 0896033929 #10544

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