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Papers on solid phase organic synthesis published in 1993

This list is arranged by the name of the first author. Any omissions, mistakes and inconsistencies please communicate to the authors of compilation (michal@5z.com). (If you are pointing to any reference, please use its ID# -- the last number in the reference.) You are welcome to use this compilation in your work. Proper way to quote it in your paper is: Lebl M., Leblova Z.: Dynamic database of references in molecular diversity. Internet http://www.5z.com.

Recently added entries are marked in bold

  1. Andrews, D.M., & Seale, P.W. (1993) Solid-phase synthesis of O-mannosylated peptides: Two strategies compared. Int. J. Peptide Prot. Res., 42, 165-170. #5845

  2. Berg, R.H., Nielsen, P.E., Buchardt, O. & Egholm, M. (1993) Peptide nucleic acids (PNA): A new strategy toward the rational design of DNA mimics. In C.H. Schneider & A.N. Eberle (Eds.), Peptides 1992, Proc.22.EPS. (pp. 152-153). ESCOM, Leiden. #4530

  3. Burdick, D.J., Struble, M.E., & Burnier, J.P. (1993) Solid phase synthesis of peptide para-nitroanilides. Tetrahedron Lett., 34, 2589-2592. #277

  4. Chen, Z.P., & Hemmasi, B. (1993) Synthesis of phytochelatins by the continuous flow solid phase procedure. Biol. Chem. Hoppe-Seyler, 374, 1057-1062. #6168

  5. Chiu, H.C., Zalipsky, S., Kopeckova, P., & Kopecek, J. (1993) Enzymatic activity of chymotrypsin and its poly(ethylene glycol) conjugates toward low and high molecular weight substrates. Bioconjug. Chem., 4, 290-295. #1377

  6. Cho, C.Y., Moran, E.J., Cherry, S.R., Stephans, J.C., Fodor, S.P.A., Adams, C.L., Sundaram, A., Jacobs, J.W., & Schultz, P.G. (1993) An unnatural biopolymer. Science, 261, 1303-1305. #478

  7. Chorev, M., & Goodman, M. (1993) A dozen years of retro-inverso peptidomimetics. Account. Chem. Res., 26, 266-273. #4526

  8. Christensen, M.K., Meldal, M., & Bock, K. (1993) Synthesis of mannose 6-phosphate-containing disaccharide threonine building blocks and their use in solid-phase glycopeptide synthesis. J. Chem. Soc. Perkin Trans. 1, 1453-1460. #1298

  9. Christiansen-Brams, I., Meldal, M., & Bock, K. (1993) Silyl protection in the solid-phase synthesis of N-linked neoglycopeptides. One-step deprotection of fully protected neoglycopeptides. Tetrahedron Lett., 34, 3315-3318. #1302

  10. Danishefsky, S.J., McCure, K.F., Randolph, J.T., & Ruggeri, R.B. (1993) A strategy for the solid-phase synthesis of oligosaccharides. Science, 260, 1307-1309. #2371

  11. DeWitt, S.H., Kiely, J.S., Stankovic, C.J., Schroeder, M.C., Cody, D.M.R., & Pavia, M.R. (1993) DIVERSOMERS: An approach to nonpeptide nonoligomeric chemical diversity. Derwent Drug File, 30, 45727-45728. #2418

  12. DeWitt, S.H., Stankovic, C.J. & Schroeder, M.C. (1993) The DIVERSOMER approach: Integration and automation of multiple, simultaneous solid phase synthesis. In J.R. Stimatitis & G.L. Hawk (Eds.), Advances in Laboratory Automation-Robotics. (pp. 248-263). Zymark Corporation, Hopkinton,MA. #2373

  13. DeWitt, S.H., Kiely, J.S., Stankovic, C.J., Schroeder, M.C., Cody, D.M.R., & Pavia, M.R. (1993) "Diversomers": An approach to nonpeptide, nonoligomeric chemical diversity. Proc. Natl. Acad. Sci. USA, 90, 6909-6913. #2372

  14. Ecker, D.J., Vickers, T.A., Hanecak, R., Driver, V., & Anderson, K. (1993) Rational screening of oligonucleotide combinatorial libraries for drug discovery. Nucl. Acid. Res., 21, 1853-1856. #668

  15. Jensen, K.J., Meldal, M., & Bock, K. (1993) Glycosylation of phenols: Preparation of 1,2-cis and 1,2-trans glycosylated tyrosine derivatives to be used in solid-phase glycopeptide synthesis. J. Chem. Soc. Perkin Trans. 1, 2119-2129. #1300

  16. Kaljuste, K., & Und n, A. (1993) New method for the synthesis of N-methyl amino acids containing peptides by reductive methylation of amino groups on the solid phase. Int. J. Peptide Prot. Res., 42, 118-124. #1172

  17. Leznoff, C.C., McArthur, C.R., & Qin, Y. (1993) Phthalocyanine-modified silica gels and their application in the purification of unsymmetrical phthalocyanines. Can. J. Chem., 71, 1319-1326. #2457

  18. Lopez, E., Chypre, C., Alpha, B., & Mathis, G. (1993) Europium (III) trisbipyridine cryptate label for time-resolved fluorescence detection of PCR products fixed on a solid support. Clin. Chem., 39, 196-201. #9967

  19. Maskos, U., & Southern, E.M. (1993) A study of oligonucleotide reassociation using large arrays of oligonucleotides synthesized on a glass support. Nucl. Acid. Res., 21, 4663-4669. #10571

  20. Mergler, M. and Nyfeler, R. Polymeric diphenyldiazomethane: A useful resin for SPPS and solid phase organic synthesis. 1993. #12541

  21. Moos, W.H., Green, G.D., & Pavia, M.R. (1993) Recent advances in the generation of molecular diversity. Annu. Rep. Med. Chem., 28, 315-324. #701

  22. Nikolaiev, V., Stierandova, A., Krchnak, V., Seligmann, B., Lam, K.S., Salmon, S.E., & Lebl, M. (1993) Peptide-encoding for structure determination of nonsequenceable polymers within libraries synthesized and tested on solid-phase supports. Peptide Res., 6, 161-170. #509

  23. Pulley, S.R., & Hegedus, L.S. (1993) Solid-phase, solution, and segment condensation peptide syntheses incorporating chromium carbene complex-derived nonproteinogenic ("unnatural") amino acid fragments. J. Amer. Chem. Soc., 115, 9037-9047. #1448

  24. Saha, A.K., Sardaro, M., Waychunas, C., Delecki, D., Kutny, R., Cavanaugh, P., Yawman, A., Upson, D.A., & Kruse, L.I. (1993) Diisopropylsilyl-linked oligonucleotide analogs: Solid-phase synthesis and physicochemical properties. J. Org. Chem., 58, 7827-7831. #5685

  25. Schwabacher, A.W., & Maynard, T.L. (1993) Preparation of peptide thioacids using the Kaiser oxime resin. Tetrahedron Lett., 34, 1269-1270. #2459

  26. Shepard, R.C. (1993) Solid-phase synthesis. Trends Biotech., 11, 492-493. #11654

  27. Smigol, V., & Svec, F. (1993) Preparation and properties of uniform beads based on macroporous glycidyl methacrylate-ethylene dimethacrylate copolymer: Use of chain transfer agent for control of the pore-size distribution. J. Appl. Polym. Sci., 48, 2033-2039. #634

  28. Smigol, V., Svec, F., & Frechet, J.M.J. (1993) Use of polymeric catalysts in the pore-size-specific functionalization of porous polymers. Macromolecules, 26, 5615-5620. #645

  29. Tamamura, H., Nakamura, J., Noguchi, K., Funakoshi, S., & Fujii, N. (1993) Acceleration of the N(alpha)-deprotection rate by the addition of m-cresol to diluted methanesulfonic acid and its application to the Z(OMe)-based solid-phase syntheses of human pancreastatin-29 and magainin-1. Chem. Pharm. Bull. Tokyo, 41, 954-957. #7837

  30. Tian, Z., Gu, C., Roeske, R.W., Zhou, M., & Van Etten, R.L. (1993) Synthesis of phosphotyrosine-containing peptides by the solid-phase method. A re-examination of the use of Boc-Tyr(PO3Bzl2)-OH. Int. J. Peptide Prot. Res., 42, 155-158. #7861

  31. Tourwe, D., Piron, J., Defreyn, P., & Van Binst, G. (1993) A new method for the solid phase synthesis of hydroxyethylamine peptide bond isosteres. Synthesis of an HIV-1 protease inhibitor and of a beta-casomorphin-5 analogue. Tetrahedron Lett., 34, 5499-5502. #7873

  32. Wenschuh, H., Beyermann, M., Krause, E., Carpino, L.A., & Bienert, M. (1993) Efficient solid phase assembly of peptides bearing contiguous highly hindered Aib residues via Fmoc Aib fluoride. Tetrahedron Lett., 34, 3733-3736. #8008

  33. Wright, P., Lloyd, D., Rapp, W., & Andrus, A. (1993) Large scale synthesis of oligonucleotides via phosphoramidite nucleosides and a high-loaded polystyrene support. Tetrahedron Lett., 34, 3373-3376. #3095

  34. Zhou, Y., & Romano, L.J. (1993) Solid-phase synthesis of oligonucleotides containing site- specific N-(2'-deoxyguanosin-8-yl)-2-(acetylamino)fluorene adducts using 9-fluorenylmethoxycarbonyl as the base-protecting group. Biochemistry, 32, 14043-14052. #706

Thursday, August 03, 2000