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Papers on solid phase organic synthesis published in 2001

This list is arranged by the name of the first author. Any omissions, mistakes and inconsistencies please communicate to the authors of compilation (michal@5z.com). (If you are pointing to any reference, please use its ID# -- the last number in the reference.) You are welcome to use this compilation in your work. Proper way to quote it in your paper is: Lebl M., Leblova Z.: Dynamic database of references in molecular diversity. Internet http://www.5z.com.

Recently added entries are marked in bold

  1. Baer, R., & Masquelin, T. (2001) A novel solid-phase approach to 2,4-diaminothiazoles. Journal of Combinatorial Chemistry, 3, 16-19. #16136

  2. Balakrishna, M.S., & Kaboudin, B. (2001) A simple and new method for the synthesis of 1,5-benzodiazepine derivatives on a solid surface. Tetrahedron Lett., 42, 1127-1129. #16416

  3. Bouloc, N., Walshe, N., & Bradley, M. (2001) Polyethers: A solid-phase iterative approach. Journal of Combinatorial Chemistry, 3, 6-8. #16134

  4. Cai, J.Q., & Wathey, B. (2001) A novel traceless solid phase tertiary amine synthesis based on Merrifield resin. Tetrahedron Lett., 42, 1383-1385. #16261

  5. Cox, P.B., Loh, V.M.Jr., Monteils, C., Baxter, A.D., & Boyd, E.A. (2001) The solid phase synthesis of unsymmetrical phosphinic acids. Tetrahedron Lett., 42, 125-128. #16229

  6. Dodd, D.S., & Zhao, Y. (2001) Solid-phase synthesis of N,N'-substituted acylguanidines. Tetrahedron Lett., 42, 1259-1262. #16274

  7. Drinnan, N., West, M.L., Broadhurst, M., Kellam, B., & Toth, I. (2001) A novel method for solid-phase synthesis of oligosaccharides using the N-1-(4,4-dimethyl-2,6-dioxocyclohexylidene)ethyl (Dde) linker. Tetrahedron Lett., 42, 1159-1162. #16279

  8. Eguchi, M., Lee, M.S., Stasiak, M., & Kahn, M. (2001) Solid-phase synthesis and solution structure of bicyclic beta-turn peptidomimetics: Diversity at the i position. Tetrahedron Lett., 42, 1237-1239. #16281

  9. Fenwick, A.E., Garnier, B., Gribble, A.D., Ife, R.J., Rawlings, A.D., & Witherington, J. (2001) Solid-phase synthesis of cyclic alkoxyketones, inhibitors of the cysteine protease cathepsin K. Bioorg. Med. Chem. Lett., 11, 195-198. #16283

  10. Galeone, A., Mayol, L., Oliviero, G., Rigano, D., & Varra, M. (2001) Solid-phase synthesis of oligonucleotides containing a bipyridine ligand at the 3'-3' inversion of polarity site. Bioorg. Med. Chem. Lett., 11, 383-386. #16287

  11. Gangloff, A.R., Litvak, J., Shelton, E.J., Sperandio, D., Wang, V.R., & Rice, K.D. (2001) Synthesis of 3,5-disubstituted-1,2,4-oxadiazoles using tetrabutylammonium fluoride as a mild and efficient catalyst. Tetrahedron Lett., 42, 1441-1443. #16418

  12. Gordon, K.H., & Balasubramanian, S. (2001) Exploring a benzyloxyaniline linker utilizing ceric ammonium nitrate (CAN) as a cleavage reagent: Solid-phase synthesis of N-unsubstituted beta-lactams and secondary amides. Organic Letters, 3, 53-56. #16292

  13. Groth, T., & Meldal, M. (2001) N-Terminal peptide aldehydes as electrophiles in combinatorial solid phase synthesis of novel peptide isosteres. Journal of Combinatorial Chemistry, 3, 45-63. #16140

  14. Groth, T., & Meldal, M. (2001) Synthesis of aldehyde building blocks protected as acid labile N-Boc N,O-acetals: Toward combinatorial solid phase synthesis of novel peptide isosteres. Journal of Combinatorial Chemistry, 3, 34-44. #16139

  15. Grotli, M., Rademan, J., Groth, T., Lubell, W.D., Miranda, L.P., & Meldal, M. (2001) Surfactant mediated cationic and anionic suspension polymerization of PEG-based resins in silicon oil: Beaded SPOCC 1500 and POEPOP 1500. Journal of Combinatorial Chemistry, 3, 28-33. #16138

  16. Gustafsson, M., Olsson, R., & Andersson, C.M. (2001) General combinatorial synthesis of tertiary amines on solid support. A novel conditional release strategy based on traceless linking at nitrogen. Tetrahedron Lett., 42, 133-136. #16230

  17. Haag, R. (2001) Dendrimers and hyperbranched polymers as high-loading supports for organic synthesis. Chem. Eur. J., 7, 327-335. #16296

  18. Hany, R., Rentsch, D., Dhanapal, B., & Obrecht, D. (2001) Quantitative determination of resin loading in solid-phase organic synthesis using 13C MAS NMR. Journal of Combinatorial Chemistry, 3, 85-89. #16145

  19. Heine, N., Germeroth, L., Schneider-Mergener, J., & Wenschuh, H. (2001) A modular approach to the SPOT synthesis of 1,3,5-trisubstituted hydantoins on cellulose membranes. Tetrahedron Lett., 42, 227-230. #16183

  20. Hone, N.D., Payne, L.J., & Tice, C.M. (2001) Direct release of nitriles from solid phase. Tetrahedron Lett., 42, 1115-1118. #16303

  21. Hwang, J.T., & Greenberg, M.M. (2001) Synthesis of 2'-modified oligodeoxynucleotides via on-column conjugation. J. Org. Chem., 66, 363-369. #16304

  22. Jin, J., Graybill, T.L., Wang, M.A., Davis, L.D., & Moore, M.L. (2001) Convenient preparation of 4-formyl-3,5-dimethoxyphenol and its incorporation into linkers and resins for solid-phase synthesis. Journal of Combinatorial Chemistry, 3, 97-101. #16147

  23. Kamal, A., Reddy, G.S.K., & Raghavan, S. (2001) Solid-phase synthesis of pyrrolo[2,1-c][1,4]benzodiazepine-5,11-diones. Bioorg. Med. Chem. Lett., 11, 387-389. #16308

  24. Kirchhoff, J.H., Brase, S., & Enders, D. (2001) A novel hydrazine linker resin and its application for the solid-phase synthesis of a-branched primary amines. Journal of Combinatorial Chemistry, 3, 71-77. #16143

  25. Kragol, G., & Otvos, L. (2001) Orthogonal solid-phase synthesis of tetramannosylated peptide constructs carrying three independent branched epitopes. Tetrahedron, 57, 957-966. #16319

  26. Lee, C.L., Chan, K.P., Lam, Y.L., & Lee, S.Y. (2001) Solid-phase combinatorial synthesis of 1,4-benzoxazin-3(4H)-one and 1,4-benzothiazin-3(4H)-one derivatives. Tetrahedron Lett., 42, 1167-1169. #16324

  27. Lee, C.L., Lam, Y., & Lee, S.Y. (2001) Solid-phase combinatorial synthesis of benzothiazole and 2,3-dihydro-[1,5]-benzothiazepine derivatives. Tetrahedron Lett., 42, 109-111. #16228

  28. Li, M., & Wilson, L.J. (2001) A facile and practical solid-phase synthesis of trisubstituted 2-aminoimidazolones. Tetrahedron Lett., 42, 1455-1458. #16420

  29. Manku, S., Laplante, C., Kopac, D., Chan, T., & Hall, D.G. (2001) A mild and general solid-phase method for the synthesis of chiral polyamines. Solution studies on the cleavage of borane-amine intermediates from the reduction of secondary amides. J. Org. Chem., 66, 874-885. #16336

  30. Marsh, A., Carlisle, S.J., & Smith, S.C. (2001) High-loading scavenger resins for combinatorial chemistry. Tetrahedron Lett., 42, 493-496. #16179

  31. Marzinzik, A. L. and Felder, E. R. Combinatorial chemistry for the identification of novel bioactive compounds. In: Anonymous. (Eds.) 1999; Wiley-VCH Verlag GmbH, Weinheim p.66 Bioorg.Chem. #16162OLD

  32. McAlpine, S.R., Lindsley, C.W., Hodges, J.C., Leonard, D.M., & Filzen, G.F. (2001) Determination of functional group distribution within Rasta resins utilizing optical analysis. Journal of Combinatorial Chemistry, 3, 1-5. #16133

  33. Meloni, M.M., & Taddei, M. (2001) Solid-phase synthesis of beta-lactams via the Miller hydroxamate approach. Organic Letters, 3, 337-340. #16340

  34. Miranda, L.P., Tao, T., Jones, A., Chernushevich, I., Standing, K.G., Geczy, C.L., & Alewood, P.F. (2001) Total chemical synthesis and chemotactic activity of human S100A12 (EN-RAGE). FEBS Lett., 488, 85-90. #16345

  35. Monnee, M.C.F., Marijne, M.F., Brouwer, A.J., & Liskamp, R.M.J. (2001) A practical solid phase synthesis of oligopeptidosulfonamide foldamers (vol 41, pg 7991, 2000). Tetrahedron Lett., 42, 965. #16346

  36. Moreno-Vargas, A.J., Fernandez-Bolanos, J.G., Fuentes, J., & Robina, I. (2001) Solution and solid phase synthesis of hetarylene-carbopeptoids. A new type of peptidomimetics. Tetrahedron Lett., 42, 1283-1285. #16348

  37. Nefzi, A., Giulianotti, M.A., & Houghten, R.A. (2001) Solid-phase synthesis of bis-heterocyclic compounds from resin-bound orthogonally protected lysine. Journal of Combinatorial Chemistry, 3, 68-70. #16142

  38. Orain, D., & Bradley, M. (2001) Solid phase synthesis of trypanothione reductase inhibitors. Towards single bead screening. Tetrahedron Lett., 42, 515-518. #16180

  39. Pattarawarapan, M., Chen, J., Steffensen, M., & Burgess, K. (2001) A rigid linker-scaffold for solid-phase synthesis of dimeric pharmacophores. Journal of Combinatorial Chemistry, 3, 102-116. #16148

  40. Piro, J., Rubiralta, M., Giralt, E., & Diez, A. (2001) Solid phase synthesis of enantiomerically pure polyhydroxyvalerolactams. Tetrahedron Lett., 42, 871-873. #16232

  41. Pirrung, M.C., & Pansare, S.V. (2001) Trityl isothiocyanate support for solid-phase synthesis. Journal of Combinatorial Chemistry, 3, 90-96. #16146

  42. Rana, S., White, P., & Bradley, M. (2001) Influence of resin cross-linking on solid-phase chemistry. Journal of Combinatorial Chemistry, 3, 9-15. #16135

  43. Reiser, U., & Jauch, J. (2001) Synthetic studies towards mniopetals (III). Solid phase organic synthesis of a key intermediate for combinatorial synthesis of mniopetals, kuehneromycins and marasmanes. Synlett, 90-92. #16367

  44. Sammelson, R.E., & Kurth, M.J. (2001) Carbon-carbon bond-forming solid-phase reactions. Part II. Chem. Rev., 101, 137-202. #16186

  45. Seneci, P. (2001) Solid-Phase Synthesis and Combinatorial Technologies. John Wiley & Sons, Inc., New York. ISBN 0471331953 #16445

  46. Tang, Q., & Wareing, J.R. (2001) Ring-closing metathesis versus cross metathesis of resin-bound olefins. Tetrahedron Lett., 42, 1399-1401. #16417

  47. Topiol, S., Davies, J., Vijayakuma, S., & Wareing, J.R. (2001) Computer aided analysis of split and mix combinatorial libraries. Journal of Combinatorial Chemistry, 3, 20-27. #16137

  48. Toy, P.H., Reger, T.S., Garibay, P., Garno, J.C., Malikayil, J.A., Liu, G., & Janda, K.D. (2001) Polytetrahydrofuran cross-linked polystyrene resins for solid-phase organic synthesis. Journal of Combinatorial Chemistry, 3, 117-124. #16149

  49. Tseng, P.H., Jiaang, W.T., Chang, M.Y., & Chen, S.T. (2001) Facile solid-phase synthesis of an antifreeze glycoprotein. Chem. Eur. J., 7, 585-590. #16397

  50. Tumelty, D., Cao, K., & Holmes, C.P. (2001) Traceless solid-phase synthesis of substituted benzimidazoles via a base-cleavable linker. Organic Letters, 3, 83-86. #16399

  51. Van Loevezijn, A., Allen, J.D., Schinkel, A.H., & Koomen, G.J. (2001) Inhibition of BCRP-mediated drug efflux by fumitremorgin-type indolyl diketopiperazines. Bioorg. Med. Chem. Lett., 11, 29-32. #16401

  52. Wang, B., Chen, L., & Kim, K. (2001) Preparation of novel 2-(trialkylsilyl)ethyl linkers and first synthesis of Tryprostatin B on solid phase. Tetrahedron Lett., 42, 1463-1466. #16421

  53. Wang, Z.G., Gu, Y.H., Zapata, A.J., & Hammond, G.B. (2001) An improved preparation of alpha-fluorinated propargylphosphonates and the solid phase synthesis of alpha-hydroxy-gamma-TIPS propargylphosphonate ester. Journal of Fluorine Chemistry, 107, 127-132. #16404

  54. Yan, B., & Yan, H. (2001) Combination of single bead FTIR and chemometrics in combinatorial chemistry: Application of the multivariate calibration method in monitoring solid-phase organic synthesis. Journal of Combinatorial Chemistry, 3, 78-84. #16144

  55. Yu, C., Jiang, Y., Liu, B., & Hu, L. (2001) A facile synthesis of 2-oxazolidinones via Hofmann rearrangement mediated by bis(trifluoroacetoxy)iodobenzene. Tetrahedron Lett., 42, 1449-1452. #16419

  56. Yu, Y., El Abdellaoui, H.M., Ostresh, J.M., & Houghten, R.A. (2001) Solid phase synthesis of [3,5,7]-1H-imidazo[1,5-a]imidazol-2(3H)-ones. Tetrahedron Lett., 42, 623-625. #16231

  57. Yun, W., Li, S., Wang, B., & Chen, L. (2001) Solid-phase synthesis of diaryl ketones through a three-component Stille coupling reaction. Tetrahedron Lett., 42, 175-177. #16182

  58. Zucca, C., Bravo, P., Volonterio, A., Zanda, M., Wagner, A., & Mioskowski, C. (2001) Regioselective solid-phase 4-amino-de-chlorination of 2,4,6-trichloropyrimidine by resin-supported N-potassium carbamates. Tetrahedron Lett., 42, 1033-1035. #16413

Tuesday, October 09, 2001