Grand
Ballroom
Town
& Country Resort & Conference Center
The fact that there is not one day dedicated to only one topic is intentional. We are trying to expose participants to different areas and we are hoping that there will be something interesting every day for everybody. We definitely don’t want chemists to come only for one day and biologists for the other. We want you all to participate, listen, talk, communicate, and most importantly, get new ideas for your research.
|
Name |
Title |
Lecture Day/Date: |
Time Slot: |
|
Schwabacher, Alan |
ONE-DIMENSIONAL SPATIAL ENCODING: SPLIT/MIX SYNTHETIC
PARALLELISM WITH TAG-FREE IDENTIFICATION AND ASSAYS AT THE SPEED OF LIGHT |
Sunday, June 10 |
8:15am - 9:00am |
|
Miranda, Les |
A NEW CONCEPT FOR THE CHEMICAL SYNTHESIS OF POLYFUNCTIONAL
MOLECULES. |
Sunday, June 10 |
9:00am - 9:20am |
|
Cavelier, Florine |
ORIGINAL AND GENERAL STRATEGY OF DIMERIZATION OF BIOACTIVE MOLECULES |
Sunday, June 10 |
9:20am - 9:40am |
|
Albericio, Fernando |
SOLID-PHASE TOTAL SYNTHESIS OF TRUNKAMIDE A AND KAHALALIDE F,
CYCLIC PEPTIDES FROM MARINE ORIGIN |
Sunday, June 10 |
9:40am - 10:00am |
|
Fields, Gregg |
TRIPLE-HELICAL PEPTIDE ANALYSIS OF COLLAGEN-OLYTIC PROTEASE
ACTIVITY |
Sunday, June 10 |
10:30am - 11:00am |
|
Garsky, Victor |
DESIGN AND SYNTHESIS OF A SELECTIVE PSA CLEAVABLE
PEPTIDE-DOXORUBICIN PRODRUG WHICH TARGETS PSA POSITIVE TUMOR CELLS. |
Sunday, June 10 |
11:00am - 11:30am |
|
Basak, Ajoy |
A HIGHLY SELECTIVE CELL PERMEABLE PEPTIDE INHIBITOR OF
PROPROTEIN CONVERTASE 1: DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION IN
CELLULAR PC1-MEDIATED PROTEOLYSIS. |
Sunday, June 10 |
11:30am - 11:50am |
|
Futaki, Shiroh |
TRANSLOCATION OF VARIOUS ARGININE-RICH PEPTIDES AND THE POTENTIAL
OF THESE PEPTIDES AS CARRIERS FOR INTRACELLULAR PROTEIN DELIVARY |
Sunday, June 10 |
11:50am - 12:10pm |
|
Vives, Eric |
NEW INSIGHTS INTO THE MEMBRANE TRANSLOCATING PROCESS OF THE TAT
PEPTIDE USED FOR CELLULAR DELIVERY OF VARIOUS BIOLOGICAL MOLECULES. |
Sunday, June 10 |
12:10pm - 12:30pm |
|
Wittmann, Valentin |
SPATIAL SCREENING OF LECTIN LIGANDS. CYCLIC PEPTIDES AS SCAFFOLDS
FOR MULTIVALENT PRESENTATION OF CARBOHYDRATES |
Sunday, June 10 |
2:30pm - 3:00pm |
|
Dunn, Ben M. |
DISCOVERIES IN PEPTIDASE SUBSTRATE SPECIFICITY: COMPARISONS
BETWEEN ANALYSIS OF SINGLE PEPTIDE SCANNING LIBRARIES AND COMBINATORIAL
LIBRARIES OF OLIGOPEPTIDES. |
Sunday, June 10 |
3:00pm - 3:20pm |
|
Slomczynska, Urszula |
COMBINATORIAL SYNTHESES OF POLYHYDROXAMATE SIDEROPHORES: DFO,
EXOCHELIN, MYCOBACTIN, AND AEORBACTIN LIBRARIES |
Sunday, June 10 |
3:20pm - 3:40pm |
|
Tegge, Werner |
DEVELOPMENT OF HIGHLY SPECIFIC, MEMRANE PERMEANT PEPTIDE
BLOCKERS OF CGMP-DEPENDENT PROTEIN KINASE UTILIZING AFFINITY SELECTION FROM
PEPTIDE LIBRARIES |
Sunday, June 10 |
3:40pm - 4:00pm |
|
Jung, Günther |
T-CELL REACTIVITY PATTERN OF PATIENTS WITH AUTOIMMUNE DISEASES
AND SUPERAGONISTS AND ANTAGONISTS FROM COMBINATORIAL LIBRARIES |
Sunday, June 10 |
4:30pm - 5:00pm |
|
Kaumaya, Pravin |
A COMBINATION OF HER-2 PEPTIDE EPITOPE VACCINES MEDIATE SUPERIOR
BIOLOGICAL EFFECTS |
Sunday, June 10 |
5:00pm - 5:30pm |
|
Lam, Kit |
IDENTIFICATION OF PEPTIDE LIGANDS FOR A4B1 INTEGRIN RECEPTOR AS
POTENTIAL TARGETING AGENTS FOR NON-HODGKIN'S LYMPHOMA |
Sunday, June 10 |
5:30pm - 6:00pm |
|
Liskamp, Rob |
COVALENT CONTROL OF SHAPE AND FOLDING IN PEPTIDES BY
RING-CLOSING METATHESIS |
Monday, June 11 |
8:00am - 8:30am |
|
Smythe, Mark |
PRIVILEGE STRUCTURES: NEW STRATEGIES FOR THE SYNTHESIS OF CYCLIC
TETRAPEPTIDES. |
Monday, June 11 |
8:30am - 8:50am |
|
Shi, Tiesheng |
A NEW REAGENT FOR THE RAPID AND QUANTITATIVE FORMATION OF
INTRAMOLECULAR DISULFIDE BONDS IN PEPTIDES |
Monday, June 11 |
8:50am - 9:10am |
|
Altstein, Miriam |
INSECT NEUROPEPTIDE ANTAGONISTS: DESIGN OF HIGHLY POTENT
INHIBITORS OF THE INSECT PHEROMONE BIOSYNTHESIS ACTIVATING NEUROPEPTIDE
(PBAN) |
Monday, June 11 |
9:10am - 9:30am |
|
Nefzi, Adel |
POLYAMINES AS INTERMEDIATES FOR THE SYNTHESIS OF HETEROCYCLIC
COMPOUNDS AND OLIGOMERIC HETEROCYCLIC COMPOUNDS FROM RESIN-BOUND POLYAMIDES |
Monday, June 11 |
9:30am - 10:00am |
|
Mosberg, Henry |
COMPARATIVE MODELING OF REMOTELY RELATED G-PROTEIN COUPLED
RECEPTORS. |
Monday, June 11 |
10:30am - 10:50am |
|
Nice, Edouard |
A TRUNCATED FORM OF THE EPIDERMAL GROWTH FACTOR RECEPTOR
ECTODOMAIN SHOWS HIGHER AFFINITY FOR EGF THAN THE FULL-LENGTH EGFR ECTODOMAIN |
Monday, June 11 |
10:50am - 11:10am |
|
Engelhard, Martin |
DESIGN AND CHEMICAL SYNTHESIS OF A PROTEIN BIOSENSOR:
INTERACTION OF THE PROTO-ONCOGENE PRODUCT H-RAS WITH THE RAS-BINDING DOMAIN
OF C-RAF 1 |
Monday, June 11 |
11:10am - 11:30am |
|
Marshall, Garland |
CONSTRAINED PEPTIDES PROBE PHOTOACTIVATED RHODOPSIN - TRANSDUCIN
INTERACTION |
Monday, June 11 |
11:30am - 12:30pm |
|
Kessler, Horst |
PEPTIDIC AND SUGAR DERIVED INHIBITORS FOR PROTEIN-PROTEIN
INTERACTION AT CELL SURFACES |
Monday, June 11 |
2:30am - 3:00pm |
|
Pessi, Antonello |
PRIME SITE BINDING INHIBITORS OF THE HEPATITIS C VIRUS NS3/4A
SERINE PROTEASE |
Monday, June 11 |
3:00pm - 3:20pm |
|
Schaschke, Norbert |
BIVALENT INHIBITION OF HUMAN BETA-TRYPTASE: PROBING THE DISTANCE
BETWEEN NEIGHBOURING SUBUNITS BY DIBASIC INHIBITORS |
Monday, June 11 |
3:20pm - 3:40pm |
|
Kiso, Yoshiaki |
PRODRUG FORMS OF PEPTIDOMIMETIC HIV PROTEASE INHIBITORS USING
INTRAMOLECULAR CYCLIZATION REACTION |
Monday, June 11 |
3:40pm - 4:00pm |
|
Naider, Fred |
PROBING THE BINDING SITE OF A HEPTAHELICAL PEPTIDE PHEROMONE
RECEPTOR USING PHOTOAFFINITY LABELLING, SITE-DIRECTED MUTAGENESIS AND
SPECTROSCOPIC APPROACHES |
Monday, June 11 |
4:30pm - 5:00pm |
|
Peggion, Evaristo |
STRUCTURE-FUNCTION RELATIONSHIP STUDIES ON ANALOGS OF THE 1-34
FRAGMENT OF PARATHYROID HORMONE (PTH) CONTAINING BETA-ALANINE RESIDUES IN
POSITIONS 11, 12 AND 13 |
Monday, June 11 |
5:00pm - 5:30pm |
|
Bracci, Luisa |
SOLUTION STRUCTURE OF THE COMPLEX OF ALPHA-BUNGAROTOXIN WITH A
MIMOTOPE OF THE ACETYLCHOLINE RECEPTOR BINDING SITE |
Monday, June 11 |
5:30pm - 5:50pm |
|
Nomizu, Motoyoshi |
CELL ATTACHMENT AND NEURITE OUTGROWTH ACTIVITIES OF LAMININ
PEPTIDE-CONJUGATED CHITOSAN MEMBRANE |
Monday, June 11 |
5:50pm - 6:10pm |
|
Seebach, Dieter |
HOMOLOGS OF AMINO ACIDS AND EXPLORATIONS INTO THE WORLDS OF
BETA- AND GAMMA- PEPTIDES |
Tuesday, June 12 |
8:00am - 8:45am |
|
Gellman, Samuel |
STRUCTURE AND FUNCTION IN BETA PEPTIDE FOLDAMERS |
Tuesday, June 12 |
8:45am - 9:30am |
|
Nowick, James |
DESIGNED AMINO ACIDS THAT INDUCE BETA-SHEET FOLDING AND
BETA-SHEET INTERACTIONS IN PEPTIDES |
Tuesday, June 12 |
9:30am - 10:00am |
|
Palian, Michael |
GLYCOPEPTIDE ANALGESICS: ALPHA HELICES AND LIPO-GLYCOPEPTIDES
WITH MORPHINE-LIKE ANALGESIA DISPLAYING REDUCED SIDE EFFECTS |
Tuesday, June 12 |
10:30am - 10:50am |
|
Otvos, Jr., Laszlo |
THE PROLINE-RICH ANTIBACTERIAL PEPTIDE FAMILY INHIBITS
CHAPERONE-ASSISTED PROTEIN FOLDING |
Tuesday, June 12 |
10:50am - 11:10am |
|
Mierke, Dale |
CHARACTERIZING THE INTERACTIONS BETWEEN CHOLECYSTOKININ AND ITS
G-PROTEIN COUPLED RECEPTOR: AN NMR-BASED STUDY |
Tuesday, June 12 |
11:10am - 11:30am |
|
Tung, Ching |
IN VIVO IMAGING OF PROTEASE ACTIVITY AND DRUG SCREENING |
Tuesday, June 12 |
11:30am - 11:50am |
|
Huang, Ziwei |
NOVEL CHEMOKINE PEPTIDES: PROBES OF LIGAND-RECEPTOR INTERACTION
AND INHIBITORS OF HIV ENTRY |
Tuesday, June 12 |
11:50am - 12:10pm |
|
Loffet, Albert |
PEPTIDES AS DRUGS: IS THERE A MARKET? |
Tuesday, June 12 |
12:10pm - 12:30pm |
|
Carter, John Mark |
A COMPREHENSIVE DATABASE OF PROTEIN-PROTEIN INTERACTIONS
INVOLVED IN INTRACELLULAR SIGNALING ACHIEVED VIA HIGH-THROUGHPUT IN VITRO
BINDING ASSAYS SUPPORTED BY HIGH-THROUGHPUT PEPTIDE SYNTHESIS. |
Wednesday, June 13 |
8:00am - 8:30am |
|
Pinilla, Clemencia |
THE INTEGRATION OF POSITIONAL SCANNING LIBRARIES WITH
BIOINFORMATICS AND PROTEOMICS |
Wednesday, June 13 |
8:30am - 9:00am |
|
Venter, Craig J. |
GENOMICS: FROM MICROBES TO MAN |
Wednesday, June 13 |
9:00am - 10:00am |
|
Gierasch, Lila |
LOCAL AND LONG-RANGE SEQUENCE CONTRIBUTIONS TO THE FOLDING OF A
PREDOMINANTLY BETA-SHEET PROTEIN |
Wednesday, June 13 |
10:30am - 11:00am |
|
Duax, William L. |
ION GATING AND SELECTIVITY IN GRAMICIDIN A |
Wednesday, June 13 |
11:00am - 11:30am |
|
Yang, Jenny J. |
CALCIUM BINDING AFFINITY AND METAL SELECTIVITY OF A DE NOVO
DESIGNED CALCIUM BINDING PROTEIN |
Wednesday, June 13 |
11:30am - 11:50am |
|
Mihara, Hisakazu |
COMPLEMENTARY ASSEMBLY OF HETEROGENEOUS MULTIPLE PEPTIDES INTO
AMYLOID FIBRILS WITH ALPHA-BETA STRUCTURAL TRANSITIONS |
Wednesday, June 13 |
11:50am - 12:10pm |
|
Lehmann, Christian |
MOLECULAR MODELING: INDISPENSABLE TOOL AT THE INTERFACE BETWEEN
STRUCTURAL ANALYSIS AND MOLECULAR DESIGN |
Wednesday, June 13 |
12:10pm - 12:30pm |
|
Schiller, Peter W. |
A GENERAL NEW CONCEPT FOR THE DEVELOPMENT OF OPIOID PEPTIDE
DERIVED MU-, DELTA- AND KAPPA-ANTAGONISTS |
Wednesday, June 13 |
2:30pm - 3:00pm |
|
Lewis, Ian |
RATIONAL APPROACH TO STABLE, UNIVERSAL SOMATOSTATIN ANALOGUES
WITH SUPERIOR THERAPEUTIC POTENTIAL |
Wednesday, June 13 |
3:00pm - 3:20pm |
|
Danho, Waleed |
HIGHLY SELECTIVE CYCLIC PEPTIDES FOR HUMAN MELANOCORTIN-4
RECEPTOR (MCR-4): DESIGN, SYNTHESIS, BIOACTIVE CONFORMATION, AND
PHARMACOLOGICAL EVALUATION AS AN ANTIOBESITY AGENT |
Wednesday, June 13 |
3:20pm - 3:40pm |
|
Haskell-Luevano, Carrie |
THE NATURALLY OCCURRING MELANOCORTIN ANTAGONIST, AGOUTI-RELATED
PROTEIN (AGRP) POSSESSES SIMILAR AND DISTINCT INTERACTIONS AT THE MC4
RECEPTOR COMPARED WITH MELANOCORTIN AGONISTS |
Wednesday, June 13 |
3:40pm - 4:00pm |
|
Giralt, Ernest |
PROLINE: A KEY BUILDING BLOCK IN PEPTIDE-BASED BIOMATERIALS |
Wednesday, June 13 |
4:30pm - 5:00pm |
|
Deber, Charles M. |
THE LYS-TAGGED PEPTIDE APPROACH TO SOLUBILIZATION OF HYDROPHOBIC
PEPTIDES. |
Wednesday, June 13 |
5:00pm - 5:30pm |
|
Lovas, Sandor |
HELIX STABILIZING AROMATIC - BACKBONE INTERACTIONS |
Wednesday, June 13 |
5:30pm - 5:50pm |
|
Yamazaki, Toshimasa |
A NEW TYPE N-TEMINAL HELIX CAPPING BOX. |
Wednesday, June 13 |
5:50pm - 6:10pm |
|
Curran, Dennis P. |
SOLID PHASE SYNTHESIS OF SMALL ORGANIC MOLECULES USING FLUOROUS
TAGGING METHODS |
Thursday, June 14 |
8:00am - 8:45am |
|
McCafferty, Dewey |
PROGRESS TOWARDS THE TOTAL SOLID-PHASE SYNTHESIS OF THE PEPTIDE
ANTIBIOTIC RAMOPLANIN A2 AGLYCONE |
Thursday, June 14 |
8:45am - 9:05am |
|
Suessmuth, Roderich D. |
SHEDDING LIGHT ON THE AGLYCON FORMATION OF GLYCOPEPTIDE
ANTIBIOTICS |
Thursday, June 14 |
9:05am - 9:25am |
|
Rapaport, Hanna |
TUNING ORDER IN B-SHEET SELF ASSEMBLY ULTRATHIN FILMS. |
Thursday, June 14 |
9:25am - 9:45am |
|
Toepert, Florian |
INCORPORATING NEW LIGAND SPECIFICITIES INTO A 38MER WW PROTEIN
DOMAIN APPLYING AN ARRAY OF 6859 WW DOMAIN VARIANTS PREPARED BY A COMBINATION
OF SPOT SYNTHESIS AND NATIVE CHEMICAL LIGATION. |
Thursday, June 14 |
9:45am - 10:05am |
|
Gras-Masse, Hélène |
HYDRAZONE LIGATION FOR THE SIMULTANEOUS LIPIDATION OF A
MULTI-EPITOPE PEPTIDE COCKTAIL |
Thursday, June 14 |
10:35am - 11:05am |
|
Andreu, David |
A DISCONTINUOUS ANTIGENIC SITE IS FUNCTIONALLY REPRODUCED BY
SYNTHETIC PEPTIDE CONSTRUCTIONS |
Thursday, June 14 |
11:05am - 11:25am |
|
Pennington, Michael |
BLOCKADE OF LYMPHOCYTE KV1.3 AND IKCA1 CHANNELS AMELIORATES
AUTOIMMUNE DEMYELINATING DISEASE IN VIVO |
Thursday, June 14 |
11:25am - 11:45am |
|
Toth, Istvan |
APPLICATIONS OF LIPOAMINO ACIDS AND LIPOSACCHARIDES FOR PEPTIDE
DELIVERY AND ENHANCING IMMUNOGENICITY |
Thursday, June 14 |
11:45am - 12:05pm |
|
Carr, Frank |
DEIMMUNISATION: A NOVEL METHOD FOR THE PRODUCTION OF THERAPEUTIC
PROTEINS WITH REDUCED IMMUNOGENICITY |
Thursday, June 14 |
12:05pm - 12:25pm |
|
Dawson, Philip |
SYNTHESIS AND CHARACTERIZATION OF PROTEINS WITH AN UNNATURAL
BACKBONE STRUCTURE OR TOPOLOGY. |
Thursday, June 14 |
2:30pm - 3:00pm |
|
Andersen, Niels |
OPTIMIZING AQUEOUS FOLD STABILITY FOR SHORT POLYPEPTIDES: A 20
RESIDUE MINIPROTEIN THAT MELTS AT 61°C |
Thursday, June 14 |
3:00pm - 3:30pm |
|
Lubell, William |
EMPLOYING THE STERIC INTERACTIONS OF 5-TERT-BUTYLPROLINE TO
CONTROL PEPTIDE FOLDING AND BIOLOGY |
Thursday, June 14 |
3:30pm - 4:00pm |
|
Offord, Robin |
PROTEIN MEDICINAL CHEMISTRY: OPTIMIZATION OF A SUPER-ACTIVE
ANTI-HIV COMPOUND. |
Thursday, June 14 |
4:30pm - 5:00pm |
|
Lipkin, Valery |
THE OCTAPEPTIDE (FRAGMENT OF DIFFERENTIATION FACTOR HLDF)
EXHIBITS NUCLEASE ACTIVITY AND INDUCES APOPTOSIS. |
Thursday, June 14 |
5:00pm - 5:20pm |
|
Tuchscherer, Gabriele |
PSEUDO-PROLINE LIBRARIES FOR TUNING INHIBITORS OF SH3 DOMAIN-MEDIATED
PROTEIN-PROTEIN INTERACTIONS |
Thursday, June 14 |
5:20pm - 5:40pm |
|
Nishiuchi, Yuji |
A COMBINED SOLID-PHASE AND SOLUTION STRATEGY FOR CHEMICAL
SYNTHESIS OF HUMAN LEPTIN |
Thursday, June 14 |
5:40pm - 6:00pm |